SCHEMBL9220670

SCHEMBL9220670

COc1cc(C(=O)NC(C)(C)C)ccc1S(=O)(=O)c1cc(Cl)cc2c1NC(=O)C2(NC(C)=O)c1ccccc1Cl

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.36
ROCK1 Q13464 2/20 0.36
HPGD P15428 1/20 0.36
CPT1A P50416 7/20 0.35
IP6K1 Q92551 1/20 0.34
PDE4D Q08499 1/20 0.34
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ACLY P53396 2/20 0.32
PTGDR Q13258 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
IMPDH2 P12268 1/20 0.32
SIRT2 Q8IXJ6 1/20 0.32
CPT1B Q92523 2/20 0.32
SCN9A Q15858 1/20 0.32
CPT2 P23786 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9218597 0.87 HPGD (0.37) ROCK2ROCK1HPGDCPT1AIP6K1
SCHEMBL9218306 0.86 ACLY (0.33) ROCK2ROCK1CPT1AACLY
SCHEMBL9212844 0.82 THRB (0.33) ROCK2ROCK1CPT1APDE4DLMNA
SCHEMBL9222097 0.80 NPSR1 (0.34) LMNATSHRACLY
SCHEMBL9219603 0.79 ACLY (0.33) ROCK2ROCK1CPT1AACLY
SCHEMBL9212102 0.79 ROCK2 (0.36) ROCK2ROCK1HPGDIP6K1PDE4D
SCHEMBL9220003 0.78 ANO1 (0.37) ROCK2ROCK1IP6K1PDE4DHDAC8
SCHEMBL7472589 0.78 AVPR1B (0.44)
SCHEMBL9221306 0.77 IDH1 (0.34) CPT1AACLY
SCHEMBL9211589 0.76 MAPT (0.37) HPGDLMNAACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0687251-A1 1,3-DIHYDROINDOL-2-ONE DERIVATIVES SUBSTITUTED IN POSITION 3 BY A NITROGEN GROUP AS VASOPRESSIN AND/OR OCYTOCINE AGONISTS AND/OR ANTAGONISTS SANOFI (FR) 1995-12-20 EP disclosed