SCHEMBL9221306

SCHEMBL9221306

CCNc1ccc(S(=O)(=O)c2cc(Cl)cc3c2NC(=O)C3(NC(=O)OC)c2ccccc2Cl)c(OC)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.34
ABCC9 O60706 1/20 0.33
ABCC8 Q09428 1/20 0.33
KCNJ11 Q14654 1/20 0.33
KCNJ8 Q15842 1/20 0.33
HTR6 P50406 1/20 0.32
TP53 P04637 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
GHSR Q92847 1/20 0.31
KDM4E B2RXH2 1/20 0.31
CCR4 P51679 3/20 0.31
GAA P10253 3/20 0.31
MAPT P10636 2/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C19 P33261 1/20 0.31
ACLY P53396 1/20 0.31
CPT1A P50416 1/20 0.31
PKLR P30613 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9217189 0.88 ABCC9 (0.34) ABCC9ABCC8KCNJ11KCNJ8TP53
SCHEMBL9219603 0.87 ACLY (0.33) GHSRGAAACLYCPT1AFABP4
SCHEMBL9211589 0.86 MAPT (0.37) HTR6TP53GHSRKDM4EGAA
SCHEMBL9217235 0.83 NPSR1 (0.35) ABCC9ABCC8KCNJ11KCNJ8TP53
SCHEMBL9217252 0.83 HTT (0.35) TP53GHSRKDM4EGAAMAPT
SCHEMBL9222097 0.82 NPSR1 (0.34) ABCC9ABCC8KCNJ11KCNJ8TP53
SCHEMBL9218306 0.80 ACLY (0.33) GHSRGAAKMT2AACLYCPT1A
SCHEMBL9218094 0.80 MAPT (0.35) ABCC9ABCC8KCNJ11KCNJ8TP53
SCHEMBL7471418 0.78 AVPR1B (0.43) IDH1MAPT
SCHEMBL9220670 0.77 ROCK2 (0.36) ACLYCPT1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0687251-A1 1,3-DIHYDROINDOL-2-ONE DERIVATIVES SUBSTITUTED IN POSITION 3 BY A NITROGEN GROUP AS VASOPRESSIN AND/OR OCYTOCINE AGONISTS AND/OR ANTAGONISTS SANOFI (FR) 1995-12-20 EP disclosed