SCHEMBL9224917

SCHEMBL9224917

CS(=O)(=O)Nc1ccc(/C=C/CN2CCN(c3ccncc3)CC2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 4/20 0.42
ADRB1 P08588 4/20 0.42
ADRB3 P13945 4/20 0.42
CYP17A1 P05093 5/20 0.41
CYP21A2 P08686 4/20 0.41
CYP11B1 P15538 4/20 0.41
KCNH2 Q12809 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP19A1 P11511 1/20 0.41
JAK2 O60674 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 3/20 0.39
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9224925 1.00 ADRB2 (0.42) ADRB2ADRB1ADRB3CYP17A1CYP21A2
SCHEMBL10680323 0.81 JAK2 (0.50) ADRB2ADRB1ADRB3KCNH2JAK2
SCHEMBL9219820 0.80 LTA4H (0.50) JAK2LMNASMN1; SMN2ALDH1A1TCF4
SCHEMBL9513748 0.80 JAK2 (0.51) ADRB2ADRB1ADRB3KCNH2CYP3A4
SCHEMBL9514747 0.78 HTR1A (0.58) KCNH2LMNASMN1; SMN2
SCHEMBL9513736 0.76 POLB (0.49) ADRB2ADRB1ADRB3KCNH2SMN1; SMN2
SCHEMBL6375438 0.75 SPHK1 (0.60) ADRB2ADRB1ADRB3KCNH2LMNA
SCHEMBL10577329 0.74 KMT2A (0.53) MEN1KMT2A
SCHEMBL9224604 0.73 SPHK1 (0.51) ADRB2ADRB1ADRB3KCNH2LMNA
SCHEMBL2022249 0.71 KCNH2 (0.78) ADRB2ADRB1ADRB3KCNH2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0484378-B1 ANTIARRHYTHMIC TERTIARY AMINE-ALKENYL-PHENYL-ALKANESULFONAMIDES UPJOHN CO (US) 1994-09-14 EP claimed
US-5405997-A Stable against rapid metabolism THE UPJOHN COMPANY (US) 1995-04-11 US disclosed
EP-0484378-B1 ANTIARRHYTHMIC TERTIARY AMINE-ALKENYL-PHENYL-ALKANESULFONAMIDES UPJOHN CO (US) 1994-09-14 EP disclosed