SCHEMBL9253837

SCHEMBL9253837

Nc1nc(N2CCOCC2)n(CN(N)C=S)n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPT P10636 1/20 0.35
PIK3CA P42336 5/20 0.33
PIK3R1 P27986 2/20 0.33
MTOR P42345 1/20 0.33
NUDT1 P36639 1/20 0.33
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
ALDH1A1 P00352 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GAA P10253 1/20 0.31
PIK3CD O00329 1/20 0.31
PIK3CB P42338 1/20 0.31
PKM P14618 1/20 0.31
AOC3 Q16853 2/20 0.30
LMNA P02545 1/20 0.30
HTT P42858 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
MAP3K12 Q12852 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9251387 0.78 GAA (0.37) CYP1A2PIK3CAPIK3R1MTORALDH1A1
SCHEMBL9248383 0.74 ALDH1A1 (0.37) ALDH1A1SMN1; SMN2
SCHEMBL9256497 0.65 CYP11B2 (0.48) PIK3CAALDH1A1SMN1; SMN2GAAPKM
SCHEMBL9843398 0.62 HRH4 (0.38)
SCHEMBL27312707 0.59 POLB (0.34) MAPTNUDT1CRHBPCRHR2ALDH1A1
SCHEMBL27312705 0.59 CRHBP (0.32) NUDT1CRHBPCRHR2
SCHEMBL9175170 0.59 ALDH1A1 (0.38) CYP1A2PIK3CAPIK3R1MTORALDH1A1
SCHEMBL9869002 0.59 ALDH1A1 (0.37) PIK3CAPIK3R1MTORALDH1A1SMN1; SMN2
SCHEMBL9257302 0.58 CA12 (0.32)
SCHEMBL21888982 0.58 AOC3 (0.41) NUDT1CRHBPCRHR2ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0425283-B1 Novel triazolyl hydrazide derivatives and process for their preparation EGYT GYOGYSZERVEGYESZETI GYAR (HU) 1995-05-10 EP disclosed
US-5225410-A Antiangina, antiulcer agents EGIS GYOGYSZERGYAR (HU) 1993-07-06 US disclosed
EP-0425283-A2 Novel triazolyl hydrazide derivatives and process for their preparation EGIS GYOGYSZERGYAR (HU) 1991-05-02 EP disclosed