SCHEMBL9254946

SCHEMBL9254946

COc1cccc2c(=O)cc(-c3ccccc3SCc3ccccc3)[nH]c12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLA P06280 1/20 0.45
GAA P10253 1/20 0.45
RAB9A P51151 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CTSB P07858 1/20 0.41
NQO2 P16083 1/20 0.41
CYP1A1 P04798 3/20 0.40
CYP1A2 P05177 3/20 0.40
CYP1B1 Q16678 3/20 0.40
MAPK3 P27361 1/20 0.40
MAPK1 P28482 1/20 0.40
MAP2K1 Q02750 1/20 0.40
MAOA P21397 1/20 0.40
ACHE P22303 1/20 0.40
MAOB P27338 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
SAE1 Q9UBE0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9258760 0.85 CYP19A1 (0.39) RAB9AL3MBTL1CTSBNQO2CYP1A1
SCHEMBL9251528 0.80 CTSV (0.46) RAB9ARXFP1MAPTKMT2ANPSR1
SCHEMBL9254180 0.79 CTSV (0.52) RAB9AMAPTKMT2ANPSR1KDM4E
SCHEMBL6534525 0.76 CYP1A1 (0.60) GLAGAANQO2CYP1A1CYP1A2
SCHEMBL9250550 0.72 KMT2A (0.57) GAARAB9ACYP1A2RXFP1MAPT
SCHEMBL3888294 0.69 L3MBTL1 (0.55) RAB9AL3MBTL1CTSBMAPTKMT2A
SCHEMBL9180770 0.69 GAA (0.58) GLAGAAL3MBTL1NQO2CYP1A1
Formaldehyde SCHEMBL28320418 0.68 RAB9A (0.51) RAB9AL3MBTL1CTSBMAPTKMT2A
SCHEMBL909732 0.68 CYP1A1 (0.56) GLAGAANQO2CYP1A1CYP1A2
SCHEMBL20605619 0.67 GAA (0.62) GLAGAAL3MBTL1NQO2CYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5393756-A Treating rheumatoid arthritis or osteoarthritis THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-02-28 US disclosed
US-5225418-A Arthritis DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1993-07-06 US disclosed