SCHEMBL9255606

SCHEMBL9255606

COc1ccc(CC(NC(=O)C(CC(=O)OCc2ccccc2)NC(=O)c2ccc3c(c2)nc(-c2ccc(C(=O)OCc4ccccc4)cc2C(=N)N)n3C)C(=O)OCc2ccccc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 3/20 0.39
F2 P00734 2/20 0.36
ERAP2 Q6P179 1/20 0.36
LNPEP Q9UIQ6 1/20 0.36
KLKB1 P03952 5/20 0.36
PTPN1 P18031 1/20 0.36
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
CTSL P07711 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
ITGB3 P05106 2/20 0.35
ITGA2B P08514 2/20 0.35
F10 P00742 1/20 0.35
ACE P12821 1/20 0.35
GPR139 Q6DWJ6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9252266 0.96 ACE (0.38) F2LNPEPKLKB1ROCK2ROCK1
SCHEMBL9252204 0.95 LNPEP (0.40) F2ERAP2LNPEPKLKB1PTPN1
SCHEMBL9252703 0.90 ENPP2 (0.39) CTSLCTSSCTSKITGB3ITGA2B
SCHEMBL9246050 0.90 HDAC6 (0.40) F2LNPEPITGB3ITGA2BF10
SCHEMBL9253897 0.87 LNPEP (0.38) F2ERAP2LNPEPCTSKITGB3
SCHEMBL9255461 0.84 HDAC6 (0.42) MMP1F2ERAP2LNPEPKLKB1
SCHEMBL9252253 0.79 HDAC6 (0.46) ACE
SCHEMBL9252518 0.75 PRSS1 (0.46) ITGB3ITGA2B
SCHEMBL9252697 0.74 HDAC6 (0.42) CTSLCTSSCTSK
SCHEMBL9246045 0.72 HDAC6 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5380729-A Treatment or prevention of neurodegenerative disorders or neurotoxic injuries STERLING WINTHROP INC. (US) 1995-01-10 US disclosed
EP-0531883-A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-03-17 EP disclosed