SCHEMBL9253897

SCHEMBL9253897

CC(C)C(NC(=O)C(CC(=O)OCc1ccccc1)NC(=O)c1ccc2c(c1)nc(-c1ccc(C(=O)OCc3ccccc3)cc1C(=N)N)n2C)C(=O)OCc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LNPEP Q9UIQ6 5/20 0.38
ERAP2 Q6P179 3/20 0.38
ERAP1 Q9NZ08 1/20 0.38
HDAC6 Q9UBN7 6/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC8 Q9BY41 1/20 0.36
CTSB P07858 1/20 0.36
CTSK P43235 1/20 0.36
PLK1 P53350 1/20 0.35
NAMPT P43490 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
KMT2A Q03164 1/20 0.35
MMP9 P14780 1/20 0.35
F10 P00742 2/20 0.34
F2 P00734 1/20 0.34
ITGB3 P05106 1/20 0.34
ITGA2B P08514 1/20 0.34
PRSS1 P07477 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9246050 0.92 HDAC6 (0.40) LNPEPHDAC6HDAC1HDAC8NAMPT
SCHEMBL9252266 0.91 ACE (0.38) LNPEPHDAC6HDAC1HDAC8NAMPT
SCHEMBL9252204 0.87 LNPEP (0.40) LNPEPERAP2ERAP1HDAC6F2
SCHEMBL9255606 0.87 MMP1 (0.39) LNPEPERAP2CTSKF10F2
SCHEMBL9252703 0.85 ENPP2 (0.39) HDAC6CTSKMEN1KMT2AITGB3
SCHEMBL9253879 0.82 HDAC6 (0.46) LNPEPERAP2ERAP1HDAC6HDAC1
SCHEMBL9252253 0.73 HDAC6 (0.46) HDAC6HDAC1HDAC8NAMPT
SCHEMBL9246045 0.73 HDAC6 (0.51) HDAC6HDAC1HDAC8NAMPT
SCHEMBL9251384 0.71 HDAC1 (0.49) HDAC6HDAC1HDAC8NAMPTF10
SCHEMBL9251561 0.70 PARP1 (0.43) ALDH1A1KMT2AF10F2PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5434150-A Anticoagulants, cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1995-07-18 US disclosed
EP-0531883-A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-03-17 EP disclosed