SCHEMBL9259482

SCHEMBL9259482

COC(=O)CCc1cn(-c2ccc(-c3ccc(C(=N)NC(=O)OC)cc3)nn2)cn1

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 2/20 0.33
NPC1 O15118 2/20 0.32
ALOX5 P09917 1/20 0.32
MAPT P10636 2/20 0.31
TP53 P04637 1/20 0.31
GAA P10253 1/20 0.31
PSEN1 P49768 1/20 0.31
PSEN2 P49810 1/20 0.31
APH1B Q8WW43 1/20 0.31
NCSTN Q92542 1/20 0.31
APH1A Q96BI3 1/20 0.31
PSENEN Q9NZ42 1/20 0.31
RAB9A P51151 1/20 0.31
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HPGD P15428 1/20 0.30
TSHR P16473 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9250749 0.92 ALOX5 (0.30) PDK1ALOX5
SCHEMBL9255212 0.91 PDK1 (0.33) PDK1NPC1MAPTTP53GAA
SCHEMBL9255067 0.89 PDK1 (0.33) PDK1NPC1ALOX5MAPTRAB9A
SCHEMBL8863938 0.89 TMPRSS15 (0.36) PDK1NPC1MAPTPSEN1PSEN2
SCHEMBL9256865 0.87 MAPT (0.33) PDK1NPC1MAPTLMNASMN1; SMN2
SCHEMBL9251525 0.83 MIF (0.37) PDK1NPC1PSEN1PSEN2APH1B
SCHEMBL9257229 0.83 SCN9A (0.38) PDK1MAPTALDH1A1LMNASMN1; SMN2
SCHEMBL8863936 0.82 CYP11B1 (0.43) PDK1NPC1MAPTALDH1A1LMNA
SCHEMBL9251800 0.82 PDK1 (0.36) PDK1NPC1MAPTTP53RAB9A
Hydrochloric Acid SCHEMBL9257352 0.82 PDK1 (0.36) PDK1NPC1MAPTRAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed