SCHEMBL9268163

SCHEMBL9268163

C1=NOc2ccccc2-c2ccccc21.NC(=O)Cl

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 4/20 0.38
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
P2RX4 Q99571 1/20 0.31
ATM Q13315 1/20 0.31
IKBKB O14920 1/20 0.31
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11830486 0.93 TRPA1 (0.35) TRPA1P2RX4ATM
Urea SCHEMBL8887503 0.93 TRPA1 (0.40) TRPA1ATMIKBKB
SCHEMBL218834 0.86 TRPA1 (0.36) TRPA1CYP1A2CYP2D6ATM
SCHEMBL9268154 0.74 KDM4E (0.33) TRPA1P2RX4ATM
SCHEMBL5944362 0.71 ALDH1A1 (0.44) TRPA1HSD17B10
SCHEMBL8804196 0.70 TRPA1 (0.36) TRPA1
SCHEMBL6173883 0.69 TRPA1 (0.39) TRPA1ATMHSD17B10
Urea SCHEMBL8887498 0.67 KDM4E (0.35) TRPA1ATM
SCHEMBL11830480 0.67 P2RX4 (0.33) P2RX4
SCHEMBL10483802 0.67 MYC (0.42) HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5449674-A Prostaglandin E2 inhibitors G. D. SEARLE & CO. (US) 1995-09-12 US disclosed
EP-0613472-A1 10-ACYL-DIBENZ(B,F) (1,4)-OXAZEPINES AND THEIR THIAZEPINES ANALO GUES USEFUL AS PROSTAGLANDIN ANTAGONISTS G.D. SEARLE & CO. (US) 1994-09-07 EP disclosed
WO-1993009104-A1 10-ACYL-DIBENZ(B,F) (1,4)-OXAZEPINES AND THEIR THIAZEPINES ANALO GUES USEFUL AS PROSTAGLANDIN ANTAGONISTS G.D. SEARLE & CO. (US) 1993-05-13 WO disclosed