SCHEMBL8804196

SCHEMBL8804196

NNC(=O)c1cccc2c1-c1ccccc1C=NO2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 4/20 0.36
CTSD P07339 2/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
ALDH1A1 P00352 3/20 0.35
P2RX7 Q99572 1/20 0.35
MYC P01106 1/20 0.34
KEAP1 Q14145 1/20 0.34
HTT P42858 1/20 0.34
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
GAA P10253 2/20 0.33
MAPT P10636 2/20 0.33
POLB P06746 1/20 0.33
MITF O75030 1/20 0.33
NCOA1 Q15788 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
NCOA3 Q9Y6Q9 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5944362 0.83 ALDH1A1 (0.44) TRPA1ALDH1A1MYCMEN1KMT2A
SCHEMBL5944439 0.77 CTSD (0.37) CTSDCA1CA2CA9ALDH1A1
Urea SCHEMBL8887503 0.72 TRPA1 (0.40) TRPA1KEAP1
SCHEMBL9268163 0.70 TRPA1 (0.38) TRPA1
SCHEMBL11830486 0.69 TRPA1 (0.35) TRPA1
SCHEMBL4779761 0.67 CTSD (0.57) CTSDCA1CA2CA9ALDH1A1
SCHEMBL541086 0.66 HNF4A (0.51) CTSDCA1CA2CA9ALDH1A1
SCHEMBL6689338 0.66 ALDH1A1 (0.64) ALDH1A1KEAP1HTTMEN1KMT2A
SCHEMBL239328 0.65 CTSD (0.63) CTSDCA1CA2CA9ALDH1A1
SCHEMBL30547074 0.65 CTSD (0.63) CTSDCA1CA2CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696283-B1 2-, 3-, 4-, 5-, 6-, 7-, 8-, 9- AND/OR 10-SUBSTITUTED DIBENZOXAZEPINE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE SEARLE & CO (US) 1997-09-17 EP disclosed