SCHEMBL9299238

SCHEMBL9299238

COc1ccc(C#CC(O)c2ccc(CN(O)C(C)=O)cc2)cc1OC

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACACB O00763 3/20 0.46
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ACHE P22303 6/20 0.41
MAPT P10636 2/20 0.41
ALDH1A1 P00352 1/20 0.41
ALOX5 P09917 2/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
LDHA P00338 1/20 0.39
BCHE P06276 3/20 0.38
PKM P14618 1/20 0.37
ALOX15 P16050 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9299121 0.88 ACACB (0.41) ACACBMEN1KMT2AACHEMAPT
SCHEMBL9299960 0.85 ACACB (0.43) ACACBMEN1KMT2AACHEMAPT
SCHEMBL9300204 0.84 PTGES (0.46) ACACBMEN1KMT2AMAPTALDH1A1
SCHEMBL9299859 0.81 ACACB (0.42) ACACBMEN1KMT2AALDH1A1ALOX5
SCHEMBL9298814 0.81 ALOX5 (0.51) ACACBMEN1KMT2AALOX5PTGS1
SCHEMBL9299666 0.80 PTGES (0.44) ALOX5PTGS1PTGS2
SCHEMBL9300259 0.79 ACHE (0.39) ACACBMEN1KMT2AACHEMAPT
SCHEMBL9299660 0.77 PTGES (0.45) ALOX5L3MBTL1
SCHEMBL9299977 0.77 ALOX5 (0.39) ALOX5PTGS1PTGS2
SCHEMBL9298923 0.76 ACHE (0.41) ACACBMEN1KMT2AACHELDHA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5326902-A Oxyalkyne compounds, pharmaceutical compositions containing them and processes for preparing such compounds and compositions GRUENENTHAL GMBH (DE) 1994-07-05 US disclosed