SCHEMBL9300259

SCHEMBL9300259

COc1ccc(C#CC(O)c2cccc(CN(O)C(N)=O)c2)cc1OC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 4/20 0.39
ACACB O00763 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.37
NR1H3 Q13133 1/20 0.37
ALDH1A1 P00352 4/20 0.37
MAPT P10636 2/20 0.37
BCHE P06276 2/20 0.36
KDM4E B2RXH2 1/20 0.36
PTGES O14684 3/20 0.36
ALOX5 P09917 2/20 0.36
LMNA P02545 2/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
HPGD P15428 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9299121 0.92 ACACB (0.41) ACHEACACBL3MBTL1NR1H3ALDH1A1
SCHEMBL9299307 0.84 ALOX5 (0.41) PTGESALOX5
SCHEMBL9299828 0.81 ALOX5 (0.36) ALOX5
SCHEMBL9299028 0.80 PTGES (0.45) KDM4EPTGESALOX5
SCHEMBL9299238 0.79 ACACB (0.46) ACHEACACBL3MBTL1ALDH1A1MAPT
SCHEMBL9299660 0.79 PTGES (0.45) L3MBTL1PTGESALOX5
SCHEMBL9300599 0.76 ALDH1A1 (0.43) L3MBTL1ALDH1A1MAPTPTGESALOX5
SCHEMBL9298923 0.76 ACHE (0.41) ACHEACACBBCHELMNAMEN1
SCHEMBL9300627 0.75 ALOX5 (0.45) PTGESALOX5MEN1KMT2A
SCHEMBL9476259 0.74 PTGES (0.58) PTGESALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5326902-A Oxyalkyne compounds, pharmaceutical compositions containing them and processes for preparing such compounds and compositions GRUENENTHAL GMBH (DE) 1994-07-05 US disclosed