SCHEMBL9299121

SCHEMBL9299121

COc1ccc(C#CC(O)c2cccc(CN(O)C(C)=O)c2)cc1OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 2/20 0.41
ALDH1A1 P00352 4/20 0.41
MAPT P10636 3/20 0.41
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ALOX5 P09917 2/20 0.38
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
ACHE P22303 3/20 0.37
BCHE P06276 2/20 0.36
KDM4E B2RXH2 1/20 0.36
PTGES O14684 3/20 0.36
LMNA P02545 2/20 0.35
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
HPGD P15428 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9300259 0.92 ACHE (0.39) ACACBALDH1A1MAPTMEN1KMT2A
SCHEMBL9299238 0.88 ACACB (0.46) ACACBALDH1A1MAPTMEN1KMT2A
SCHEMBL9300627 0.84 ALOX5 (0.45) MEN1KMT2AALOX5PTGS1PTGS2
SCHEMBL9299727 0.81 FFAR1 (0.38) ALOX5PTGS1PTGS2
SCHEMBL9300204 0.77 PTGES (0.46) ACACBALDH1A1MAPTMEN1KMT2A
SCHEMBL9299960 0.76 ACACB (0.43) ACACBALDH1A1MAPTMEN1KMT2A
SCHEMBL9299307 0.75 ALOX5 (0.41) ALOX5PTGES
SCHEMBL9299666 0.73 PTGES (0.44) ALOX5PTGS1PTGS2PTGES
SCHEMBL9197316 0.72 PTGES (0.59) ACACBALOX5PTGS1PTGS2PTGES
SCHEMBL9299828 0.72 ALOX5 (0.36) ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5326902-A Oxyalkyne compounds, pharmaceutical compositions containing them and processes for preparing such compounds and compositions GRUENENTHAL GMBH (DE) 1994-07-05 US disclosed