SCHEMBL9300560

SCHEMBL9300560

CC(=O)N(O)Cc1ccc(C(O)C#Cc2ccccn2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.44
PTGS1 P23219 1/20 0.44
PTGS2 P35354 1/20 0.44
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
PKM P14618 1/20 0.42
HPGD P15428 1/20 0.42
HTT P42858 1/20 0.42
ATM Q13315 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
FFAR1 O14842 1/20 0.40
HSD17B2 P37059 1/20 0.36
PTGES O14684 1/20 0.36
AKR1C3 P42330 1/20 0.36
GAA P10253 1/20 0.34
GRM5 P41594 3/20 0.34
PPARD Q03181 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9298814 0.83 ALOX5 (0.51) ALOX5PTGS1PTGS2FFAR1PTGES
SCHEMBL9299806 0.79 ALOX5 (0.41) ALOX5PTGS1PTGS2ALDH1A1NPSR1
SCHEMBL9299128 0.78 FFAR1 (0.43) ALOX5PTGS1PTGS2FFAR1PTGES
SCHEMBL9299975 0.77 ACACB (0.43) ALOX5PTGS1PTGS2GRM5
SCHEMBL9299899 0.76 ALOX5 (0.39) ALOX5PTGS1PTGS2ALDH1A1HPGD
SCHEMBL9300599 0.76 ALDH1A1 (0.43) ALOX5ALDH1A1MAPTPKMHPGD
SCHEMBL9299859 0.76 ACACB (0.42) ALOX5PTGS1PTGS2ALDH1A1HTT
SCHEMBL9300204 0.75 PTGES (0.46) ALOX5PTGS1PTGS2ALDH1A1MAPT
SCHEMBL9299666 0.74 PTGES (0.44) ALOX5PTGS1PTGS2PTGESAKR1C3
SCHEMBL9299977 0.74 ALOX5 (0.39) ALOX5PTGS1PTGS2FFAR1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5326902-A Oxyalkyne compounds, pharmaceutical compositions containing them and processes for preparing such compounds and compositions GRUENENTHAL GMBH (DE) 1994-07-05 US disclosed