SCHEMBL9301516

SCHEMBL9301516

CC(C)(C)OC(=O)C1CCCN1c1cc2c(cc1F)n1c(=O)[nH]c(=O)cc1n2C1CC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.34
ATR Q13535 1/20 0.33
ATRIP Q8WXE1 1/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC8 Q9BY41 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
GABRG2 P18507 2/20 0.32
GABRB3 P28472 2/20 0.32
GABRA5 P31644 2/20 0.32
GABRA4 P48169 2/20 0.32
GABRA6 Q16445 2/20 0.32
GPR174 Q9BXC1 1/20 0.31
ALDH1A1 P00352 3/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
TRPV1 Q8NER1 1/20 0.31
HRH3 Q9Y5N1 4/20 0.30
OPRM1 P35372 1/20 0.30
OPRD1 P41143 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9303487 0.84 HDAC1 (0.34) CASP3ATRATRIPHDAC1HDAC8
SCHEMBL9304073 0.81 MAPT (0.39) ALDH1A1HRH3OPRM1OPRD1OGFRL1
SCHEMBL9303648 0.78 ACE (0.34) CASP3TRPV1OPRM1OPRD1OPRK1
SCHEMBL9302040 0.75 KDM4E (0.41) ALDH1A1CYP2C9
SCHEMBL9301517 0.73 CASP3 (0.33) CASP3ROCK2
SCHEMBL9847716 0.71 HDAC1 (0.36) ATRATRIPHDAC1HDAC8HDAC6
SCHEMBL9301818 0.71 ATR (0.35) ATRATRIPHDAC1HDAC8HDAC6
SCHEMBL9303841 0.69 HPGD (0.35) ATRATRIPHDAC1HDAC8HDAC6
SCHEMBL9302272 0.66 MAPT (0.42) GPR174ALDH1A1CYP2C9CYP2C19
SCHEMBL9301295 0.64 OPRM1 (0.36) ALDH1A1HRH3OPRM1OPRD1OGFRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5283248-A Bactericides, enzyme inhibitor of DNA-gyrase in bacteria HOFFMANN-LA ROCHE INC. (US) 1994-02-01 US disclosed