SCHEMBL9847716

SCHEMBL9847716

CC(C)(C)OC(=O)C1CCCN1c1cc2c(cc1F)nc(CC(=O)O)n2C1CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.36
HDAC8 Q9BY41 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
ATR Q13535 1/20 0.35
ATRIP Q8WXE1 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
OGFRL1 Q5TC84 1/20 0.34
CYP11B2 P19099 6/20 0.33
CYP11B1 P15538 5/20 0.33
CYP19A1 P11511 1/20 0.33
RORC P51449 1/20 0.33
CREBBP Q92793 1/20 0.33
CPT1A P50416 1/20 0.33
GPR174 Q9BXC1 1/20 0.32
JAK2 O60674 1/20 0.32
JAK1 P23458 1/20 0.32
TYK2 P29597 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9301818 0.92 ATR (0.35) HDAC1HDAC8HDAC6ATRATRIP
SCHEMBL9303841 0.91 HPGD (0.35) HDAC1HDAC8HDAC6ATRATRIP
SCHEMBL9303690 0.85 OPRM1 (0.37) HDAC1HDAC8HDAC6ATRATRIP
SCHEMBL9847732 0.81 HTT (0.43) OPRM1OPRD1OGFRL1CYP11B2CYP11B1
SCHEMBL9847728 0.80 OGFRL1 (0.38) OPRM1OPRD1OPRK1OGFRL1CYP11B2
SCHEMBL9301681 0.73 HTT (0.42) OPRM1OPRD1OGFRL1CYP11B2CYP11B1
SCHEMBL9301682 0.72 RORC (0.42) OPRM1OPRD1OGFRL1CYP11B2CYP11B1
SCHEMBL9301581 0.72 HTT (0.50) OPRM1OPRD1OGFRL1CYP11B2CYP11B1
SCHEMBL9301471 0.72 RORC (0.41) OPRM1OPRD1OGFRL1CYP11B2CYP11B1
SCHEMBL9303487 0.71 HDAC1 (0.34) HDAC1HDAC8HDAC6ATRATRIP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0433648-A1 Substituted pyrimidobenzimidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1991-06-26 EP disclosed