SCHEMBL9302147

SCHEMBL9302147

CCn1c(C(N)=S)nc2cc(F)c(N3CCN(C)CC3)cc21

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.41
RAD52 P43351 1/20 0.41
DRD3 P35462 1/20 0.41
KDM4E B2RXH2 5/20 0.38
ALDH1A1 P00352 3/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
NPC1 O15118 1/20 0.38
HPGD P15428 1/20 0.38
CSF1R P07333 2/20 0.38
OPRL1 P41146 1/20 0.38
GLA P06280 1/20 0.37
HTT P42858 1/20 0.36
LMNA P02545 1/20 0.36
SOS1 Q07889 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9303256 0.80 GAA (0.45) GAARAD52DRD3KDM4EALDH1A1
SCHEMBL9847719 0.76 DRD3 (0.47) GAARAD52DRD3KDM4EALDH1A1
SCHEMBL9301127 0.75 DRD3 (0.39) GAARAD52DRD3KDM4EALDH1A1
SCHEMBL9302130 0.73 HTT (0.47) GAARAD52DRD3KDM4EALDH1A1
SCHEMBL9847735 0.70 HTT (0.43) GAARAD52DRD3KDM4EALDH1A1
SCHEMBL9303370 0.69 ALDH1A1 (0.43) GAARAD52DRD3KDM4EALDH1A1
SCHEMBL6803657 0.68 DRD3 (0.53) GAARAD52DRD3KDM4EALDH1A1
SCHEMBL9302311 0.68 CYP11B2 (0.44) GAARAD52DRD3KDM4EALDH1A1
Hydrochloric Acid SCHEMBL9302957 0.67 CYP11B1 (0.43) GAARAD52DRD3KDM4EALDH1A1
SCHEMBL9302880 0.66 HTT (0.46) GAAKDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5283248-A Bactericides, enzyme inhibitor of DNA-gyrase in bacteria HOFFMANN-LA ROCHE INC. (US) 1994-02-01 US disclosed
EP-0433648-A1 Substituted pyrimidobenzimidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1991-06-26 EP disclosed