SCHEMBL9303370

SCHEMBL9303370

CCn1c(CC(=O)NOCc2ccccc2)nc2cc(F)c(N3CCN(C)CC3)cc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.43
KDM4E B2RXH2 6/20 0.43
HPGD P15428 2/20 0.43
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
LMNA P02545 2/20 0.41
GAA P10253 3/20 0.39
RAD52 P43351 1/20 0.39
DRD3 P35462 2/20 0.39
USP2 O75604 1/20 0.39
NOD2 Q9HC29 1/20 0.39
NPC1 O15118 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
RAB9A P51151 1/20 0.38
GRM5 P41594 1/20 0.38
TSHR P16473 1/20 0.37
CSF1R P07333 2/20 0.36
HSD17B10 Q99714 2/20 0.36
ALOX15 P16050 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9302144 0.87 GRM5 (0.39) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL9847719 0.81 DRD3 (0.47) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL9303256 0.81 GAA (0.45) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL9301969 0.78 GRM5 (0.42) ALDH1A1HPGDKMT2ALMNASMN1; SMN2
SCHEMBL9302130 0.78 HTT (0.47) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL9302252 0.76 ACHE (0.42) LMNAGRM5
SCHEMBL9847735 0.73 HTT (0.43) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL9301127 0.71 DRD3 (0.39) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL9302880 0.70 HTT (0.46) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL9302147 0.69 GAA (0.41) ALDH1A1KDM4EHPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5283248-A Bactericides, enzyme inhibitor of DNA-gyrase in bacteria HOFFMANN-LA ROCHE INC. (US) 1994-02-01 US disclosed
EP-0433648-A1 Substituted pyrimidobenzimidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1991-06-26 EP disclosed