SCHEMBL9847719

SCHEMBL9847719

CCn1c(CC(=O)O)nc2cc(F)c(N3CCN(C)CC3)cc21

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 1/20 0.47
KDM4E B2RXH2 8/20 0.44
ALDH1A1 P00352 6/20 0.44
MEN1 O00255 6/20 0.44
KMT2A Q03164 6/20 0.44
HPGD P15428 2/20 0.44
NPC1 O15118 1/20 0.44
GAA P10253 2/20 0.43
RAD52 P43351 1/20 0.43
HTT P42858 1/20 0.40
GLA P06280 1/20 0.40
LMNA P02545 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9303256 0.90 GAA (0.45) DRD3KDM4EALDH1A1MEN1KMT2A
SCHEMBL9302130 0.87 HTT (0.47) DRD3KDM4EALDH1A1MEN1KMT2A
SCHEMBL9847735 0.82 HTT (0.43) DRD3KDM4EALDH1A1MEN1KMT2A
SCHEMBL9303370 0.81 ALDH1A1 (0.43) DRD3KDM4EALDH1A1MEN1KMT2A
SCHEMBL9301127 0.81 DRD3 (0.39) DRD3KDM4EALDH1A1MEN1KMT2A
SCHEMBL9302147 0.76 GAA (0.41) DRD3KDM4EALDH1A1MEN1KMT2A
SCHEMBL9302880 0.76 HTT (0.46) KDM4EALDH1A1MEN1KMT2AHPGD
Acetic Acid SCHEMBL9301936 0.75 CYP11B2 (0.44) DRD3KDM4EALDH1A1MEN1KMT2A
SCHEMBL9302311 0.73 CYP11B2 (0.44) DRD3KDM4EALDH1A1MEN1KMT2A
SCHEMBL9301930 0.73 HTT (0.45) DRD3KDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0433648-A1 Substituted pyrimidobenzimidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1991-06-26 EP disclosed