SCHEMBL9302494

SCHEMBL9302494

c1ccc2c(c1)OC(CNCC1CCNCC1)CS2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 9/20 0.49
TP53 P04637 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
TSHR P16473 1/20 0.49
CYP2C19 P33261 1/20 0.49
HIF1A Q16665 1/20 0.49
MEN1 O00255 1/20 0.48
PMP22 Q01453 1/20 0.48
KMT2A Q03164 1/20 0.48
ADRA1D P25100 8/20 0.42
ADRA1B P35368 8/20 0.42
NISCH Q9Y2I1 1/20 0.40
PRMT5 O14744 1/20 0.39
WDR77 Q9BQA1 1/20 0.39
KDM1A O60341 2/20 0.36
MAOB P27338 2/20 0.36
MAOA P21397 1/20 0.36
CHRM1 P11229 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9302556 0.77 ADRA1D (0.65) ADRA1AADRA1DADRA1B
SCHEMBL6097642 0.76 ADRA1A (0.45) ADRA1ATP53CYP1A2CYP3A4CYP2D6
SCHEMBL9302459 0.74 CXCR4 (0.54) ADRA1ATP53CYP1A2CYP3A4CYP2D6
SCHEMBL9301885 0.73 CXCR4 (0.56) ADRA1ATP53CYP1A2CYP3A4CYP2D6
SCHEMBL9302550 0.71 ADRA1A (0.53) ADRA1ATP53CYP1A2CYP3A4CYP2D6
SCHEMBL11638248 0.71 ADRA1A (0.44) ADRA1ATP53CYP1A2CYP3A4CYP2D6
SCHEMBL9301904 0.70 ADRA1A (0.51) ADRA1ATP53CYP1A2CYP3A4CYP2D6
SCHEMBL14367858 0.66 ADRA1A (0.51) ADRA1ATP53CYP1A2CYP3A4CYP2D6
SCHEMBL11222841 0.66 ADRA1A (0.43) ADRA1ATP53CYP1A2CYP3A4CYP2D6
SCHEMBL14367876 0.66 ADRA1A (0.51) ADRA1ATP53CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5286735-A Antidepressants, anxiolytic agents PIERRE FABRE MEDICAMENT (FR) 1994-02-15 US claimed
US-5286735-A Antidepressants, anxiolytic agents PIERRE FABRE MEDICAMENT (FR) 1994-02-15 US disclosed