SCHEMBL9302550

SCHEMBL9302550

COc1cccc(CN2CCC(CNCC3CSc4ccccc4O3)CC2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 3/20 0.53
ADRA1D P25100 2/20 0.53
ADRA1B P35368 2/20 0.53
ACHE P22303 5/20 0.49
BACE1 P56817 2/20 0.49
SIGMAR1 Q99720 2/20 0.49
TP53 P04637 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
TSHR P16473 1/20 0.48
CYP2C19 P33261 1/20 0.48
HIF1A Q16665 1/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
PMP22 Q01453 1/20 0.48
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 2/20 0.45
MAPT P10636 1/20 0.45
DRD4 P21917 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9301885 0.88 CXCR4 (0.56) ADRA1AACHEBACE1TP53CYP1A2
SCHEMBL9302459 0.87 CXCR4 (0.54) ADRA1AADRA1DADRA1BSIGMAR1TP53
SCHEMBL9301600 0.84 ADRA1D (0.74) ADRA1AADRA1DADRA1BMEN1KMT2A
SCHEMBL9301904 0.82 ADRA1A (0.51) ADRA1AADRA1DADRA1BTP53CYP1A2
SCHEMBL9302546 0.78 SIGMAR1 (0.46) SIGMAR1KDM4EALDH1A1MAPTDRD4
SCHEMBL7375679 0.72 SIGMAR1 (0.65) ACHESIGMAR1KDM4EALDH1A1MAPT
SCHEMBL9302364 0.72 EPHX2 (0.46) ADRA1ATP53CYP1A2CYP3A4CYP2D6
SCHEMBL9302823 0.71 ADRA1D (0.62) ADRA1AADRA1DADRA1BSIGMAR1KDM4E
SCHEMBL9303150 0.71 ADRA1D (0.59) ADRA1AADRA1DADRA1BSIGMAR1ALDH1A1
SCHEMBL9300949 0.71 ADRA1D (0.66) ADRA1AADRA1DADRA1BACHEBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5286735-A Antidepressants, anxiolytic agents PIERRE FABRE MEDICAMENT (FR) 1994-02-15 US claimed
US-5286735-A Antidepressants, anxiolytic agents PIERRE FABRE MEDICAMENT (FR) 1994-02-15 US disclosed