SCHEMBL9302845

SCHEMBL9302845

N=C(N)Nc1cccc(C(=O)Nc2ccc(C(=N)N)c3ccccc23)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.52
CLK1 P49759 1/20 0.46
SIRT2 Q8IXJ6 2/20 0.45
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
AKR1C4 P17516 1/20 0.44
AKR1C3 P42330 1/20 0.44
AKR1C2 P52895 1/20 0.44
AKR1C1 Q04828 1/20 0.44
KCNK3 O14649 2/20 0.43
KCNK9 Q9NPC2 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
PLAU P00749 2/20 0.43
F2 P00734 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9303308 0.94 PTGES (0.56) PTGESCLK1SIRT2NPC1RAB9A
SCHEMBL9303113 0.86 CD40 (0.51) SIRT2NPC1RAB9ACYP1A2CYP3A4
SCHEMBL9304048 0.85 SIRT2 (0.55) PTGESSIRT2KCNK3KCNK9MEN1
SCHEMBL9303515 0.82 PTGES (0.48) PTGESNPC1RAB9AMEN1KMT2A
SCHEMBL9302930 0.82 PTGES (0.51) PTGESSIRT2NPC1RAB9ACYP1A2
SCHEMBL9304320 0.81 PLAU (0.50) PTGESSIRT2NPC1RAB9AKCNK3
SCHEMBL9303405 0.81 NPC1 (0.48) SIRT2NPC1RAB9ACYP1A2CYP3A4
SCHEMBL7501198 0.80 PKM (0.48) PTGESCLK1NPC1RAB9ACYP1A2
SCHEMBL9302840 0.80 PTGES (0.51) PTGESSIRT2NPC1RAB9AKCNK3
SCHEMBL9304163 0.80 PTGES (0.54) PTGESNPC1RAB9ACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5352704-A Antiviral agents BANYU PHARMACEUTICAL CO., LTD. (JP) 1994-10-04 US disclosed
EP-0434432-B1 Guanidinobenzene derivatives BANYU PHARMA CO LTD (JP) 1994-05-04 EP disclosed
EP-0434432-A1 Guanidinobenzene derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 1991-06-26 EP disclosed