SCHEMBL9304657

SCHEMBL9304657

NCCn1nc(-c2ccc(C(F)(F)F)cc2)c2cnccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.41
SRC P12931 2/20 0.39
BRAF P15056 2/20 0.39
KDR P35968 2/20 0.39
MAPK14 Q16539 2/20 0.39
AXL P30530 1/20 0.37
TYRO3 Q06418 1/20 0.37
MERTK Q12866 1/20 0.37
NAMPT P43490 1/20 0.37
SCN9A Q15858 4/20 0.37
MAOB P27338 1/20 0.36
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
TYK2 P29597 1/20 0.35
JAK3 P52333 1/20 0.35
SMO Q99835 1/20 0.35
KCNH2 Q12809 1/20 0.34
KDM4E B2RXH2 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MAPK13 O15264 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9305227 0.93 KIF11 (0.40) KIF11SRCBRAFKDRMAPK14
SCHEMBL9304368 0.91 MERTK (0.39) KIF11SRCBRAFKDRMAPK14
Maleic Acid SCHEMBL8143988 0.90 FTO (0.40) KIF11NAMPTSCN9AJAK2JAK1
Fumaric Acid SCHEMBL8143990 0.90 FTO (0.40) KIF11NAMPTSCN9AJAK2JAK1
SCHEMBL9258008 0.88 NAMPT (0.39) MAPK14MERTKNAMPTMAOBKDM4E
SCHEMBL9302703 0.83 CSNK2A2 (0.39) SRCBRAFKDRNAMPTKCNH2
SCHEMBL8137072 0.83 ALDH1A1 (0.39) NAMPTMAOBKDM4ENPSR1
SCHEMBL9306122 0.82 HSD17B10 (0.47) MERTKMAOBKDM4E
Hydrochloric Acid SCHEMBL8134231 0.81 HSD17B10 (0.46) MERTKMAOBKDM4E
SCHEMBL9304792 0.80 MAPK13 (0.41) BRAFMAPK14MERTKNAMPTMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5296491-A Pyrazolo[4,3-c]pyridines and their use as serotonin reuptake inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-22 US claimed