Fumaric Acid

Fumaric Acid

SCHEMBL9304831

CC(C)Oc1ccccc1N1CCN(Cc2ccc(C(=O)N3CCCCC3)s2)CC1.O=C(O)C=CC(=O)O

nearest known ligand 0.89

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ATP4AATP4BAXLBTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CHRM2CHRM3CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4FLT3HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3KCNH2KMT2AMAP2K1MAP2K2MEN1MLNRMPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PLK4PPARGRENS1PR1SLC6A2SLC6A3SLC6A4SMOTYK2atpAatpBatpCatpDatpEatpFatpFHatpGpol

The experimentally established mechanism targets of Fumaric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADRA1D known ✓ P25100 2/20 0.60
ADRA1A known ✓ P35348 2/20 0.60
ADRA1B known ✓ P35368 2/20 0.60
HTR1A known ✓ P08908 1/20 0.60
DRD2 known ✓ P14416 1/20 0.60
HTR1B P28222 1/20 0.60
DRD3 P35462 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL9304827 1.00 ADRA1D (0.60) ADRA1DADRA1AADRA1BHTR1ADRD2
SCHEMBL9305919 0.94 ADRA1D (0.66) ADRA1DADRA1AADRA1BHTR1ADRD2
SCHEMBL9305535 0.94 ADRA1D (0.66) ADRA1DADRA1AADRA1BHTR1ADRD2
Hydrochloric Acid SCHEMBL9307647 0.94 ADRA1D (0.65) ADRA1DADRA1AADRA1BHTR1ADRD2
SCHEMBL9305702 0.79 ADRA1D (0.70) ADRA1DADRA1AADRA1BHTR1ADRD2
SCHEMBL9305855 0.79 ADRA1D (0.70) ADRA1DADRA1AADRA1BHTR1ADRD2
Hydrochloric Acid SCHEMBL9304961 0.78 ADRA1D (0.69) ADRA1DADRA1AADRA1BHTR1ADRD2
SCHEMBL7646052 0.77 HTR1A (0.68) ADRA1DADRA1AADRA1BHTR1ADRD2
SCHEMBL9539641 0.77 HTR1A (0.80) ADRA1DADRA1AADRA1BHTR1ADRD2
Hydrochloric Acid SCHEMBL7648139 0.76 HTR1A (0.79) ADRA1DADRA1AADRA1BHTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5332732-A Thiophene and pyridine antipsychotic agents MCNEILAB, INC. (US) 1994-07-26 US disclosed