SCHEMBL9308466

SCHEMBL9308466

CNc1ccc(C(=O)Cl)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.45
RECQL P46063 2/20 0.45
HSD17B10 Q99714 2/20 0.45
TP53 P04637 2/20 0.45
HIF1A Q16665 2/20 0.45
CYP3A4 P08684 1/20 0.45
THRB P10828 1/20 0.45
HPGD P15428 1/20 0.45
ALOX15 P16050 1/20 0.45
CASP1 P29466 1/20 0.45
HDAC3 O15379 2/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC2 Q92769 2/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
TSHR P16473 1/20 0.40
APP P05067 3/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5745396 0.90 KCNQ3 (0.46) ALDH1A1CA1CA2NPC1RAB9A
SCHEMBL4140392 0.80 CES2 (0.52) ALDH1A1RECQLHSD17B10TP53HIF1A
SCHEMBL11596462 0.80 MAPK13 (0.52) ALDH1A1HSD17B10THRBHPGDALOX15
SCHEMBL52136 0.80 ALDH1A1 (0.52) ALDH1A1RECQLHSD17B10TP53HIF1A
SCHEMBL20587670 0.79 ALDH1A1 (0.59) ALDH1A1TP53HPGDALOX15CA12
SCHEMBL68148 0.79 ALDH1A1 (0.59) ALDH1A1TP53HPGDALOX15CA12
SCHEMBL912761 0.78 KMT2A (0.56) ALDH1A1TP53HPGDCA12CA1
SCHEMBL18724447 0.78 ALDH1A1 (0.45) ALDH1A1HSD17B10TP53HIF1AHDAC1
SCHEMBL98312 0.78 TSHR (0.60) ALDH1A1TP53HPGDALOX15CA12
SCHEMBL64499 0.77 ALDH1A1 (0.63) ALDH1A1HSD17B10TP53HIF1ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100372838-C Piperidine-benzenesulfonamide derivatives HOFFMANN LA ROCHE (CH) 2008-03-05 CN disclosed
CN-1751023-A Piperidine-benzenesulfonamide derivatives HOFFMANN LA ROCHE (CH) 2006-03-22 CN disclosed
US-5332735-A Antiamnesic activity ADIR ET COMPAGNIE (FR) 1994-07-26 US disclosed
US-4155905-A 6-Substituted penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1979-05-22 US disclosed
US-4077967-A 6-Substituted penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1978-03-07 US disclosed
US-4069224-A N-(PYRIDYLALKYL)BENZAMIDES, IMPROVE PRODUCTION OF PROSTAGLANDINS IN MAMMALS THE UPJOHN COMPANY (US) 1978-01-17 US disclosed
US-4061851-A 7-Amino-7-arylthio cephalosporins E. R. SQUIBB & SONS, INC. (US) 1977-12-06 US disclosed
US-4061629-A 6-Amino-6-arylthio penicillanic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1977-12-06 US disclosed
US-4029669-A 6-Benzalimino-6-arylthio penicillanic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1977-06-14 US disclosed
US-4026886-A 7-Acyl-7-arylthiocephalosporins E. R. SQUIBB & SONS, INC. (US) 1977-05-31 US disclosed
US-3965093-A 6-Arylthio penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1976-06-22 US disclosed
US-3954744-A ANTIBACTERIAL E. R. SQUIBB & SONS, INC. (US) 1976-05-04 US disclosed