SCHEMBL9320730

SCHEMBL9320730

O=CNCCc1cc(O)cc(O)c1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.43
CBS P35520 1/20 0.41
PTGS2 P35354 3/20 0.41
CYP3A4 P08684 1/20 0.41
ACHE P22303 1/20 0.39
HSP90AB1 P08238 1/20 0.38
TYR P14679 1/20 0.37
ADRB2 P07550 2/20 0.37
LMNA P02545 1/20 0.37
ADH1B P00325 1/20 0.34
ADH1A P07327 1/20 0.34
ADH7 P40394 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9320706 0.81 DRD2 (0.52) CYP3A4
SCHEMBL2701814 0.79 TMEM97 (0.55) ADRB2LMNA
SCHEMBL28157468 0.76 CBS (0.50) LTA4HCBSPTGS2CYP3A4ACHE
SCHEMBL6652052 0.75 CNR1 (0.44) CYP3A4LMNAADH1BADH1AADH7
SCHEMBL8763412 0.75 LMNA (0.50) LMNAADH1BADH1AADH7
SCHEMBL6815570 0.75 MAPT (0.59) PTGS2CYP3A4ACHEADRB2LMNA
SCHEMBL31076394 0.75 MAPT (0.59) PTGS2CYP3A4ACHEADRB2LMNA
SCHEMBL5361823 0.72 LMNA (0.36) PTGS2ACHEADRB2LMNAADH1B
SCHEMBL13093762 0.71 TMEM97 (0.61) LTA4HPTGS2CYP3A4ACHELMNA
SCHEMBL10149325 0.71 LTA4H (0.74) LTA4HCBSPTGS2CYP3A4ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0440887-B1 Improvement in the total synthesis of Erbstatin analogs ERBA CARLO SPA (IT) 1994-01-26 EP disclosed
US-5130472-A TOTAL SYNTHESIS OF ERBSTATIN ANALOGS FARMITALIA CARLO ERBA S.R.L. (IT) 1992-07-14 US disclosed
EP-0440887-A1 Improvement in the total synthesis of Erbstatin analogs FARMITALIA CARLO ERBA S.r.l. (IT) 1991-08-14 EP disclosed