SCHEMBL932329

SCHEMBL932329

O=CC(Oc1ccccc1)N1CCN(S(=O)(=O)c2ccc3ncsc3c2)CC1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.49
CHRM5 P08912 3/20 0.44
RAB9A P51151 2/20 0.44
MAPT P10636 2/20 0.44
KDM4E B2RXH2 1/20 0.44
NAMPT P43490 1/20 0.42
NPC1 O15118 1/20 0.40
IKBKB O14920 5/20 0.40
ALDH1A1 P00352 4/20 0.39
HPGD P15428 2/20 0.39
CHUK O15111 3/20 0.38
VDR P11473 1/20 0.38
GFER P55789 1/20 0.38
GPR55 Q9Y2T6 1/20 0.38
PKM P14618 1/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL932971 0.80 MCOLN3 (0.58) ALDH1A1PKMHTT
SCHEMBL932636 0.79 ALDH1A1 (0.50) ALDH1A1PKM
SCHEMBL931510 0.77 PKM (0.59) KDM4EALDH1A1HPGDPKMHTT
SCHEMBL9950422 0.76 PKM (0.64) MAPTKDM4EALDH1A1PKMHTT
SCHEMBL932795 0.76 LMNA (0.42) GBA1KDM4EPKMHTT
SCHEMBL933278 0.72 KMT2A (0.54) MAPTALDH1A1PKMHTT
SCHEMBL932990 0.72 PKM (0.62) ALDH1A1PKMHTT
SCHEMBL932085 0.72 SMN1; SMN2 (0.55) MAPTPKMHTT
SCHEMBL8414638 0.71 IKBKB (0.60) GBA1CHRM5RAB9AMAPTKDM4E
SCHEMBL28013845 0.71 RAB9A (0.67) GBA1CHRM5RAB9AMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2448581-A1 THERAPEUTIC COMPOSITIONS AND RELATED METHODS OF USE Agios Pharmaceuticals, Inc. (US) 2012-05-09 EP disclosed
WO-2011002816-A1 THERAPEUTIC COMPOSITIONS AND RELATED METHODS OF USE AGIOS PHARMACEUTICALS, INC. (US) 2011-01-06 WO disclosed