SCHEMBL9324701

SCHEMBL9324701

O=C(O)NN1CC=C(c2cccc3ccccc23)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 2/20 0.47
HTR1D P28221 3/20 0.41
HTR1B P28222 3/20 0.41
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
GAA P10253 2/20 0.39
HTR6 P50406 2/20 0.38
HTT P42858 1/20 0.38
MAPT P10636 1/20 0.37
HDAC8 Q9BY41 2/20 0.37
HTR2C P28335 1/20 0.37
NPC1 O15118 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6711077 0.82 ALDH1A1 (0.56) ALDH1A1KDM4EHTR1DHTR1BLMNA
SCHEMBL9323906 0.75 HTR1A (0.49) KDM4E
SCHEMBL7255363 0.73 HTR6 (0.58) KDM4ELMNAPOLBHTR6ALOX15
SCHEMBL9674614 0.73 HTR1D (0.45) ALDH1A1KDM4EHTR1DHTR1BGAA
SCHEMBL7957307 0.72 HTR1D (0.51) HTR1DHTR1BHTR6
Bromide SCHEMBL9325716 0.72 HTR6 (0.57) KDM4ELMNAPOLBHTR6ALOX15
SCHEMBL6042752 0.70 DRD2 (0.63) KDM4EGAAHTR6HTTMAPT
SCHEMBL7957405 0.70 TNF (0.50) HTR1DHTR1B
SCHEMBL6847847 0.70 PDK4 (0.69) HTR6
SCHEMBL9031902 0.68 HTR1D (0.50) HTR1DHTR1BGAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5292761-A Piperidine, tetrahydropyridine and pyrrolidine compounds ADIR ET COMPAGNIE (FR) 1994-03-08 US disclosed
US-5260317-A Hypotensive agents ADIR ET COMPAGNIE (FR) 1993-11-09 US disclosed
US-5250544-A Hypotensive agents ADIR ET COMPAGNIE (FR) 1993-10-05 US disclosed
US-5240942-A Hypotensive agents; 5-hydroxytryptamine antagonist ADIR ET COMPAGNIE (FR) 1993-08-31 US disclosed