SCHEMBL9340684

SCHEMBL9340684

COC(=O)Cc1cccc(O[Si](C)(C)C(C)(C)C)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.44
DRD2 P14416 1/20 0.41
ALDH1A1 P00352 2/20 0.41
GAA P10253 1/20 0.41
GFER P55789 1/20 0.41
CTBP2 P56545 1/20 0.41
HSP90AB1 P08238 2/20 0.41
POLB P06746 2/20 0.40
GLS O94925 1/20 0.40
HSP90AA1 P07900 1/20 0.40
RAB9A P51151 2/20 0.39
SYK P43405 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PDK2 Q15119 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3235704 0.87 CYP1A2 (0.49) CTBP2HSP90AB1HSP90AA1
SCHEMBL4190201 0.86 DRD2 (0.50) SMN1; SMN2DRD2HSP90AB1POLBHSP90AA1
SCHEMBL18294034 0.85 AOC2 (0.47) ALDH1A1HSP90AB1POLBGLSHSP90AA1
SCHEMBL6362544 0.84 F10 (0.44) DRD2CTBP2HSP90AB1HSP90AA1
SCHEMBL1279084 0.84 MEN1 (0.46) SMN1; SMN2ALDH1A1POLBMAPTHPGD
SCHEMBL14987130 0.83 SLC7A5 (0.41) SLC7A5SMN1; SMN2ALDH1A1GAAGLS
SCHEMBL3839217 0.82 CYP4F2 (0.50) SMN1; SMN2DRD2ALDH1A1GAAGFER
SCHEMBL10196989 0.82 F10 (0.44) DRD2CTBP2HSP90AB1GLSHSP90AA1
SCHEMBL4183069 0.82 HSP90AB1 (0.61) SMN1; SMN2DRD2ALDH1A1GAAGFER
SCHEMBL10697163 0.81 HSP90AA1 (0.41) DRD2ALDH1A1CTBP2HSP90AB1GLS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12516055-B2 Protein kinase inhibitors and uses thereof for the treatment of diseases and conditions TRUSTEES OF TUFTS COLLEGE (US) 2026-01-06 US disclosed
EP-4480485-A2 PROTEIN KINASE INHIBITORS AND USES THEREOF FOR THE TREATMENT OF DISEASES AND CONDITIONS University of Houston System (US) 2024-12-25 EP disclosed
EP-3968991-B1 PROTEIN KINASE INHIBITORS AND USES THEREOF FOR THE TREATMENT OF DISEASES AND CONDITIONS UNIV HOUSTON SYSTEM (US) 2024-07-31 EP disclosed
EP-4276092-A1 COMPOUND LIBRARY CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2023-11-15 EP disclosed
EP-4276092-A1 COMPOUND LIBRARY CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2023-11-15 EP disclosed
US-11708347-B2 Substituted benzofuran, benzopyrrole, benzothiophene, and structurally related complement inhibitors BIOCRYST PHARMACEUTICALS, INC. (US) 2023-07-25 US disclosed
US-20220194937-A1 PROTEIN KINASE INHIBITORS AND USES THEREOF FOR THE TREATMENT OF DISEASES AND CONDITIONS UNIVERSITY OF HOUSTON SYSTEM 2022-06-23 US disclosed
EP-3968991-A1 PROTEIN KINASE INHIBITORS AND USES THEREOF FOR THE TREATMENT OF DISEASES AND CONDITIONS University of Houston System (US) 2022-03-23 EP disclosed
WO-2020232190-A1 PROTEIN KINASE INHIBITORS AND USES THEREOF FOR THE TREATMENT OF DISEASES AND CONDITIONS UNIVERSITY OF HOUSTON SYSTEM (US) 2020-11-19 WO disclosed
US-5362879-A 4-5-diphenyloxazole derivatives as inhibitors of blood platelet aggregation BRISTOL-MYERS SQUIBB COMPANY (US) 1994-11-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220194937-A1 PROTEIN KINASE INHIBITORS AND USES THEREOF FOR THE TREATMENT OF DISEASES AND CONDITIONS RIPK2, RIPK1, RIPK4 SLC7A5 4269/4885SMN1; SMN2 1451/4885DRD2 4421/4885
US-11708347-B2 Substituted benzofuran, benzopyrrole, benzothiophene, and structurally related complement inhibitors C9, C5, C1QBP SLC7A5 2191/4885SMN1; SMN2 2080/4885DRD2 4071/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.