SCHEMBL9341809

SCHEMBL9341809

OC1(c2ccccn2)CCCc2ccc(C(F)(F)C(F)(F)F)cc21

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 3/20 0.35
TRPV3 Q8NET8 1/20 0.34
PDK2 Q15119 2/20 0.34
NR3C1 P04150 5/20 0.33
CYP11B1 P15538 3/20 0.33
CYP11B2 P19099 3/20 0.33
CYP17A1 P05093 2/20 0.33
CYP3A4 P08684 2/20 0.33
SIGMAR1 Q99720 1/20 0.33
SYK P43405 1/20 0.33
TMEM97 Q5BJF2 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2B Q13224 1/20 0.32
BRD4 O60885 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
OPRK1 P41145 1/20 0.31
OPRL1 P41146 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9340020 0.81 HSD11B1 (0.36) HSD11B1TRPV3PDK2CYP11B1CYP11B2
SCHEMBL9340819 0.79 APP (0.40) PDK2CYP11B1CYP11B2CYP17A1CYP3A4
SCHEMBL9339909 0.76 TRPV3 (0.41) TRPV3NR3C1CYP11B1CYP11B2CYP17A1
SCHEMBL8315208 0.71 TRPV3 (0.35) HSD11B1TRPV3PDK2
SCHEMBL6902549 0.70 SIGMAR1 (0.43) PDK2SIGMAR1GRIN1GRIN2AGRIN2B
SCHEMBL8126674 0.70 CYP3A4 (0.47) CYP11B1CYP11B2CYP17A1CYP3A4SIGMAR1
SCHEMBL15467881 0.63 TRPV1 (0.37) HSD11B1CYP11B1CYP11B2CYP17A1CYP3A4
SCHEMBL8312787 0.61 TRPV3 (0.43) HSD11B1TRPV3PDK2
SCHEMBL768782 0.60 AKR1B1 (0.40) SIGMAR1
SCHEMBL29730766 0.60 GRIN1 (0.51) HSD11B1PDK2GRIN1GRIN2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5356915-A Antihypertensive and bronchodilator agents J. URIACH & CIA. S.A. (ES) 1994-10-18 US disclosed
EP-0600147-A1 Tetralones with pharmacological activity, compositions containing them and process for their preparation J. URIACH & CIA. S.A. (ES) 1994-06-08 EP disclosed