SCHEMBL9339909

SCHEMBL9339909

OC1(c2ccccn2)CCCc2cc(Cl)c(Cl)cc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV3 Q8NET8 1/20 0.41
CYP3A4 P08684 3/20 0.36
CYP11B1 P15538 3/20 0.36
CYP11B2 P19099 3/20 0.36
CYP17A1 P05093 2/20 0.36
NR3C1 P04150 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2A Q12879 1/20 0.35
GRIN2B Q13224 1/20 0.35
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
OPRL1 P41146 1/20 0.34
KDM1A O60341 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9340819 0.81 APP (0.40) CYP3A4CYP11B1CYP11B2CYP17A1GRIN1
SCHEMBL8126674 0.77 CYP3A4 (0.47) CYP3A4CYP11B1CYP11B2CYP17A1KDM1A
SCHEMBL9341796 0.76 HSD11B1 (0.37) TRPV3GRIN1GRIN2AGRIN2BOPRM1
SCHEMBL9341809 0.76 HSD11B1 (0.35) TRPV3CYP3A4CYP11B1CYP11B2CYP17A1
SCHEMBL6902549 0.72 SIGMAR1 (0.43) GRIN1GRIN2AGRIN2BOPRM1OPRD1
SCHEMBL8313558 0.67 SLC6A2 (0.38) TRPV3NR3C1OPRM1OPRL1CHRM2
SCHEMBL8311725 0.64 SLC6A2 (0.36) NR3C1
SCHEMBL29980976 0.64 OPRM1 (0.57) GRIN1GRIN2AGRIN2BOPRM1OPRD1
SCHEMBL536677 0.64 OPRM1 (0.57) GRIN1GRIN2AGRIN2BOPRM1OPRD1
SCHEMBL29980665 0.64 OPRM1 (0.57) GRIN1GRIN2AGRIN2BOPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5356915-A Antihypertensive and bronchodilator agents J. URIACH & CIA. S.A. (ES) 1994-10-18 US disclosed
EP-0600147-A1 Tetralones with pharmacological activity, compositions containing them and process for their preparation J. URIACH & CIA. S.A. (ES) 1994-06-08 EP disclosed