Fumaric Acid

Fumaric Acid

SCHEMBL9345641

CN1CCC(NC(=O)C(C)(C)CO[N+](=O)[O-])CC1.O=C(O)C=CC(=O)O

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ATP4AATP4BAXLBTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CHRM2CHRM3CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4FLT3HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3KCNH2KMT2AMAP2K1MAP2K2MEN1MLNRMPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PLK4PPARGRENS1PR1SLC6A2SLC6A3SLC6A4SMOTYK2atpAatpBatpCatpDatpEatpFatpFHatpGpol

The experimentally established mechanism targets of Fumaric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 20/20 0.54
SSTR1 P30872 7/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9329945 0.93 SSTR4 (0.57) SSTR4SSTR1
SCHEMBL9346132 0.80 SSTR4 (0.43) SSTR4SSTR1
Fumaric Acid SCHEMBL9348870 0.77 LMNA (0.41) SSTR4
SCHEMBL9329974 0.76 SSTR4 (0.52) SSTR4SSTR1
Fumaric Acid SCHEMBL9348823 0.76 LMNA (0.40)
SCHEMBL9345695 0.74 SSTR4 (0.62) SSTR4SSTR1
Fumaric Acid SCHEMBL9348961 0.74 MMP2 (0.38)
SCHEMBL9329832 0.73 SSTR4 (0.45) SSTR4SSTR1
SCHEMBL9329969 0.71 SSTR4 (0.57) SSTR4SSTR1
Fumaric Acid SCHEMBL9795190 0.70 BCHE (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5280031-A Cyclic azaaliphatic compounds with a nitroxy function, processes for the preparation thereof and pharmaceutical compositions containing them BOEHRINGER MANNHEIM GMBH (DE) 1994-01-18 US disclosed
US-5030641-A Treatment of angina pectoris, hypotensive agents BOEHRINGER MANNHEIM GMBH (DE) 1991-07-09 US disclosed