SCHEMBL9358982

SCHEMBL9358982

Cc1cc2c(-c3ccccc3Cl)c(NC(=O)Nc3ccccc3)c(=O)n(C)c2cc1C

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.47
FPR2 P25090 7/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
TACR1 P25103 1/20 0.45
MAPT P10636 2/20 0.45
POLB P06746 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
LMNA P02545 1/20 0.44
ALDH1A1 P00352 1/20 0.43
RAB9A P51151 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
WEE1 P30291 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9363075 0.94 FPR2 (0.53) PKMFPR2L3MBTL1SMN1; SMN2MAPT
SCHEMBL9363416 0.92 TACR1 (0.54) PKMFPR2SMN1; SMN2TACR1MAPT
SCHEMBL9359119 0.92 PKM (0.56) PKMFPR2L3MBTL1SMN1; SMN2TACR1
SCHEMBL9363425 0.88 KDR (0.51) PKMFPR2MAPTMEN1KMT2A
SCHEMBL9359288 0.87 DDX3X (0.49) PKMSMN1; SMN2MAPTPOLBMEN1
SCHEMBL7642011 0.85 HTT (0.45) SMN1; SMN2RAB9A
SCHEMBL9359046 0.84 MAPT (0.41) FPR2SMN1; SMN2MAPTPOLBMEN1
SCHEMBL9358730 0.80 LMNA (0.44) L3MBTL1TACR1POLBMEN1KMT2A
SCHEMBL9358719 0.77 LMNA (0.50) PKMTACR1MAPTPOLBMEN1
SCHEMBL6634344 0.77 ROCK2 (0.41) MAPTLMNAWEE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0421456-B1 Quinoline derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1994-12-28 EP disclosed
US-5223513-A Anticholesterol agent TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-06-29 US disclosed
EP-0421456-A2 Quinoline derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-04-10 EP disclosed