SCHEMBL9364872

SCHEMBL9364872

CC(C)[C@H](N)C(=O)N(NC(=O)OCc1ccccc1)[C@@H](CCCc1ccccc1)[C@H]1OC(C)(C)O[C@@H]1[C@H](CCCc1ccccc1)N(NC(=O)OCc1ccccc1)C(=O)[C@@H](N)C(C)C

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 4/20 0.38
MMP8 P22894 1/20 0.37
MMP14 P50281 1/20 0.37
SLC15A1 P46059 1/20 0.37
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
SLC1A3 P43003 1/20 0.36
SLC1A1 P43005 1/20 0.36
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
CASP1 P29466 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ATM Q13315 1/20 0.36
ERAP2 Q6P179 1/20 0.36
ERAP1 Q9NZ08 1/20 0.36
LNPEP Q9UIQ6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9364447 0.93 LNPEP (0.40) NAAASLC15A1ALDH1A1CYP3A4TSHR
SCHEMBL9699796 0.81 CTSK (0.41) NAAAALDH1A1CYP3A4TSHRSLC1A3
SCHEMBL9699824 0.76 SLC15A1 (0.41) NAAASLC15A1ALDH1A1SLC1A3SLC1A1
SCHEMBL9369693 0.73 CTSL (0.44) SLC15A1SLC1A3SLC1A1CTSLCTSB
SCHEMBL7476658 0.73 SLC15A1 (0.46) SLC15A1SLC1A3SLC1A1CTSLCTSB
SCHEMBL9364548 0.72 CTSK (0.45) SLC15A1SLC1A3SLC1A1CTSLCTSB
SCHEMBL9364449 0.68 SLC15A1 (0.45) MMP8MMP14SLC15A1ALDH1A1
SCHEMBL7324719 0.65 SLC15A1 (0.53) SLC15A1ALDH1A1CTSLCTSBCTSS
SCHEMBL7324724 0.65 SLC15A1 (0.53) SLC15A1ALDH1A1CTSLCTSBCTSS
SCHEMBL966186 0.65 HTT (0.55) ALDH1A1SLC1A3SLC1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0538396-A4 1994-04-13 EP disclosed
EP-0538396-A1 INHIBITORS OF RETROVIRAL PROTEASES SMITHKLINE BEECHAM CORPORATION (US) 1993-04-28 EP disclosed
WO-1992000948-A1 INHIBITORS OF RETROVIRAL PROTEASES SMITHKLINE BEECHAM CORPORATION (US) 1992-01-23 WO disclosed