SCHEMBL9364447

SCHEMBL9364447

CCCC[C@@H]([C@H]1OC(C)(C)O[C@@H]1[C@H](CCCC)N(NC(=O)OCc1ccccc1)C(=O)[C@@H](N)C(C)C)N(NC(=O)OCc1ccccc1)C(=O)[C@@H](N)C(C)C

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LNPEP Q9UIQ6 2/20 0.40
CTSL P07711 2/20 0.40
CTSS P25774 2/20 0.40
ERAP2 Q6P179 1/20 0.38
SLC15A1 P46059 1/20 0.37
NAAA Q02083 2/20 0.37
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
SLC1A3 P43003 1/20 0.36
SLC1A1 P43005 1/20 0.36
CTSB P07858 1/20 0.36
CTSK P43235 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9364872 0.93 NAAA (0.38) LNPEPCTSLCTSSERAP2SLC15A1
SCHEMBL9699796 0.81 CTSK (0.41) CTSLCTSSNAAAALDH1A1CYP3A4
SCHEMBL9369693 0.81 CTSL (0.44) LNPEPCTSLCTSSERAP2SLC15A1
SCHEMBL9699824 0.76 SLC15A1 (0.41) CTSLCTSSSLC15A1NAAAALDH1A1
SCHEMBL7476658 0.73 SLC15A1 (0.46) CTSLCTSSSLC15A1SLC1A3SLC1A1
SCHEMBL9364548 0.72 CTSK (0.45) CTSLCTSSSLC15A1SLC1A3SLC1A1
SCHEMBL9012148 0.69 CTSB (0.44) CTSLCTSSCYP3A4CTSBCTSK
SCHEMBL5501379 0.67 CTSL (0.61) CTSLCTSSCTSBCTSK
SCHEMBL7266217 0.67 ALDH1A1 (0.52) LNPEPCTSLCTSSERAP2ALDH1A1
SCHEMBL7266221 0.67 ALDH1A1 (0.52) LNPEPCTSLCTSSERAP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0538396-A4 1994-04-13 EP disclosed
EP-0538396-A1 INHIBITORS OF RETROVIRAL PROTEASES SMITHKLINE BEECHAM CORPORATION (US) 1993-04-28 EP disclosed
WO-1992000948-A1 INHIBITORS OF RETROVIRAL PROTEASES SMITHKLINE BEECHAM CORPORATION (US) 1992-01-23 WO disclosed