SCHEMBL9397274

SCHEMBL9397274

O=S(=O)(c1ccc(Cl)c2ncccc12)N1CCNCC1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.64
NFKB1 P19838 3/20 0.64
TSHR P16473 2/20 0.64
THPO P40225 1/20 0.64
HIF1A Q16665 1/20 0.64
LMNA P02545 4/20 0.63
MAPT P10636 3/20 0.63
BLM P54132 1/20 0.63
COMT P21964 4/20 0.59
KDM4E B2RXH2 2/20 0.57
CYP1A2 P05177 3/20 0.54
CYP2D6 P10635 3/20 0.54
MYLK Q15746 3/20 0.54
MAPK1 P28482 2/20 0.54
TP53 P04637 2/20 0.54
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
CYP2C9 P11712 1/20 0.54
GMNN O75496 2/20 0.53
PMP22 Q01453 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9397148 0.95 CYP3A4 (0.62) CYP3A4NFKB1TSHRTHPOHIF1A
SCHEMBL17962258 0.87 COMT (0.78) CYP3A4NFKB1TSHRTHPOHIF1A
SCHEMBL9397169 0.81 ALDH1A1 (0.72) CYP3A4NFKB1TSHRTHPOHIF1A
SCHEMBL29968116 0.78 CYP3A4 (1.00) CYP3A4NFKB1TSHRTHPOHIF1A
SCHEMBL9397276 0.78 CYP3A4 (1.00) CYP3A4NFKB1TSHRTHPOHIF1A
SCHEMBL9397241 0.78 FTO (0.43) CYP3A4NFKB1TSHRTHPOHIF1A
SCHEMBL9397232 0.78 TSHR (0.53) CYP3A4NFKB1TSHRTHPOHIF1A
SCHEMBL9397254 0.77 ALDH1A1 (0.67) CYP3A4NFKB1TSHRTHPOHIF1A
SCHEMBL2712002 0.77 L3MBTL1 (0.71) CYP3A4NFKB1TSHRTHPOHIF1A
SCHEMBL2908180 0.76 ROCK2 (0.67) CYP3A4NFKB1TSHRTHPOHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5340811-A Bronchodilator agent ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1994-08-23 US disclosed
EP-0471841-A1 SULFONAMIDE DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1992-02-26 EP disclosed