SCHEMBL9397299

SCHEMBL9397299

CC(NS(=O)(=O)c1cccc2ncccc12)N1CCCNCC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.56
NFKB1 P19838 3/20 0.56
TSHR P16473 2/20 0.56
THPO P40225 1/20 0.56
HIF1A Q16665 1/20 0.56
LMNA P02545 3/20 0.55
MAPT P10636 3/20 0.55
BLM P54132 1/20 0.55
HTR1A P08908 3/20 0.41
HTR6 P50406 2/20 0.41
HTR7 P34969 2/20 0.41
DRD2 P14416 1/20 0.41
ROCK1 Q13464 5/20 0.41
ROCK2 O75116 4/20 0.41
PRKX P51817 2/20 0.41
PRKCE Q02156 2/20 0.41
PRKCD Q05655 2/20 0.41
PRKD1 Q15139 2/20 0.41
CCKBR P32239 1/20 0.40
CYP2D6 P10635 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9397252 0.83 FTO (0.40) CYP3A4NFKB1TSHRTHPOHIF1A
SCHEMBL9398259 0.80 PRKD3 (0.61) CYP3A4NFKB1TSHRTHPOHIF1A
SCHEMBL9397241 0.78 FTO (0.43) CYP3A4NFKB1TSHRTHPOHIF1A
SCHEMBL16000113 0.78 LMNA (0.50) CYP3A4NFKB1TSHRTHPOHIF1A
SCHEMBL9398471 0.75 CYP3A4 (0.90) CYP3A4NFKB1TSHRTHPOHIF1A
SCHEMBL9397203 0.75 PRKD3 (0.61) CYP3A4NFKB1TSHRTHPOHIF1A
SCHEMBL9397301 0.75 TSHR (0.57) CYP3A4NFKB1TSHRTHPOHIF1A
SCHEMBL9398247 0.75 ALDH1A1 (0.54) CYP3A4LMNAMAPTCYP2D6CYP2C19
SCHEMBL9349827 0.74 HTR1A (0.51) HTR1AHTR6HTR7DRD2KCNH2
SCHEMBL9397253 0.73 MAPK1 (0.51) CYP3A4NFKB1LMNAHTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5340811-A Bronchodilator agent ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1994-08-23 US disclosed
EP-0471841-A1 SULFONAMIDE DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1992-02-26 EP disclosed