SCHEMBL9399794

SCHEMBL9399794

CC(C)(C)OC(=O)N1CCC([C@@H]2C[C@H](SC(c3ccccc3)(c3ccccc3)c3ccccc3)CN2C(=O)OCc2ccc([N+](=O)[O-])cc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 6/20 0.48
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
GPR119 Q8TDV5 1/20 0.40
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
HTT P42858 1/20 0.39
AGTR2 P50052 1/20 0.38
ATM Q13315 1/20 0.38
PARP1 P09874 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9399880 0.91 CCR5 (0.49) CCR5TDP1AGTR2ATMRAB9A
SCHEMBL9020939 0.83 CCR5 (0.44) CCR5ALDH1A1LMNAMAPTGPR119
SCHEMBL7860693 0.81 TDP1 (0.43) CCR5ALDH1A1TDP1ATMNPC1
SCHEMBL9363103 0.81 MGLL (0.41) CCR5ALDH1A1TDP1ATMPARP1
SCHEMBL9399205 0.80 CCR5 (0.45) CCR5ALDH1A1LMNAMAPTGPR119
SCHEMBL9020004 0.80 CCR5 (0.41) CCR5ALDH1A1LMNAMAPTTDP1
SCHEMBL9399096 0.80 ALDH1A1 (0.43) CCR5ALDH1A1LMNAMAPTGPR119
SCHEMBL7805543 0.79 TDP1 (0.43) CCR5ALDH1A1MAPTTDP1ATM
SCHEMBL9363174 0.79 CCR5 (0.42) CCR5TDP1ATM
SCHEMBL9366889 0.79 CCR5 (0.44) CCR5JAK2JAK1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5374720-A A thienamycins bactericides has nontoxic, side effect reduction against the kidney and central nervous system BANYU PHARMACEUTICAL CO., LTD. (JP) 1994-12-20 US disclosed