Luzindole

Luzindole

SCHEMBL4869000

CC(=O)NCCc1c(Cc2ccccc2)[nH]c2ccccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 10/20 1.00
MTNR1B P49286 10/20 1.00
CYP1A2 P05177 4/20 1.00
CYP2C19 P33261 4/20 1.00
CYP3A4 P08684 3/20 1.00
HPGD P15428 3/20 1.00
TSHR P16473 3/20 1.00
TDP1 Q9NUW8 3/20 1.00
MEN1 O00255 2/20 1.00
CYP2C9 P11712 2/20 1.00
KMT2A Q03164 2/20 1.00
ALDH1A1 P00352 2/20 0.71
CYP2D6 P10635 2/20 0.71
MAPT P10636 2/20 0.71
ALOX15 P16050 2/20 0.71
CHRNB2 P17787 1/20 0.51
CHRNA7 P36544 1/20 0.51
CHRNA4 P43681 1/20 0.51
KDM4E B2RXH2 1/20 0.50
HSD17B10 Q99714 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9401161 0.91 MTNR1A (0.84) MTNR1AMTNR1BCYP1A2CYP2C19CYP3A4
Luzindole SCHEMBL9118261 0.90 MEN1 (0.81) MTNR1AMTNR1BCYP1A2CYP2C19CYP3A4
SCHEMBL9751553 0.88 MTNR1A (0.79) MTNR1AMTNR1BCYP1A2CYP2C19CYP3A4
SCHEMBL9401112 0.88 MTNR1A (0.79) MTNR1AMTNR1BCYP1A2CYP2C19CYP3A4
SCHEMBL9302251 0.87 MTNR1A (0.77) MTNR1AMTNR1BCYP1A2CYP2C19CYP3A4
SCHEMBL9304093 0.86 MTNR1A (0.75) MTNR1AMTNR1BCYP1A2CYP2C19CYP3A4
SCHEMBL9304037 0.84 MTNR1A (1.00) MTNR1AMTNR1BCYP1A2CYP2C19CYP3A4
SCHEMBL9303475 0.84 MTNR1A (0.72) MTNR1AMTNR1BCYP1A2CYP2C19CYP3A4
SCHEMBL1626901 0.83 MTNR1A (1.00) MTNR1AMTNR1BCYP1A2CYP2C19CYP3A4
SCHEMBL9302872 0.83 MTNR1A (0.71) MTNR1AMTNR1BCYP1A2CYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 73 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5283343-A Melatonin antagonists WHITBY RESEARCH, INC. (US) 1994-02-01 US claimed
JP-4173777-A None JP disclosed
EP-4618962-A2 METHODS AND COMPOSITIONS FOR TREATING CANCER Onconova Therapeutics, Inc. (US) 2025-09-24 EP disclosed
EP-4551578-A1 MACROCYCLIC INHIBITORS OF KRAS FOR THE TREATMENT OF CANCER F. Hoffmann-La Roche AG (CH) 2025-05-14 EP disclosed
EP-4532503-A1 HALOINDOLE MACROCYCLIC COMPOUNDS FOR THE TREATMENT OF CANCER F. Hoffmann-La Roche AG (CH) 2025-04-09 EP disclosed
EP-4526289-A1 ANTIVIRAL INDOLINYL COMPOUNDS AND USES THEREOF GILEAD SCIENCES, INC. (US) 2025-03-26 EP disclosed
EP-4502609-A2 DETERMINING A CIRCADIAN RHYTHM Vanda Pharmaceuticals Inc. (US) 2025-02-05 EP disclosed
US-12201604-B2 Treatment of circadian rhythm disorders VANDA PHARMACEUTICALS INC. (US) 2025-01-21 US disclosed
WO-2024259241-A1 5-HT2A RECEPTOR MODULATORS AND METHODS OF USE THEREOF Transneural Therapeutics, Inc. (US) 2024-12-19 WO disclosed
EP-4444300-A2 INHIBITORS OF MENIN-MLL INTERACTION Bala Therapeutics, Inc. (US) 2024-10-16 EP disclosed
EP-0549916-A2 Compounds useful as antiproliferative agents WHITBY RESEARCH, Inc. (US) 1993-07-07 EP disclosed
US-5206377-A Compounds useful as antiproliferative agents WHITBY RESEARCH, INC. (US) 1993-04-27 US disclosed
US-5151446-A Neurological disorders or cardiovascular disorders NORTHWESTERN UNIVERSITY (US) 1992-09-29 US disclosed
JP-H04173777-A MELATONINE ANALOGUE WHITBY RES INC 1992-06-22 JP disclosed
US-5093352-A Melatonin inhibitor, sleep, 2-aryl N-acetyl tryptamine WHITBY RESEARCH, INC. (US) 1992-03-03 US disclosed
US-5071875-A Nervous system, psychological disorders; sleep cycle, skin dis coloration NORTHWESTERN UNIVERSITY (US) 1991-12-10 US disclosed
EP-0420064-A2 Substituted 2-amidotetralins as melatonin agonists and antagonists NORTHWESTERN UNIVERSITY (US) 1991-04-03 EP disclosed
EP-0375726-A4 MELATONIN ANALOGUES 1991-01-30 EP disclosed
EP-0375726-A1 MELATONIN ANALOGUES Whitby Research Incorporated (US) 1990-07-04 EP disclosed
WO-1989001472-A1 MELATONIN ANALOGUES NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-02-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12201604-B2 Treatment of circadian rhythm disorders CRY1, PER2, CRY2 MTNR1A 4/4885MTNR1B 5/4885CYP1A2 256/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.