SCHEMBL9402298

SCHEMBL9402298

COC(N)=S.Cc1ccc(-c2ccccc2C(=O)OC(C)(C)C)cc1.NC(O)=S

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 4/20 0.46
SLC6A4 P31645 3/20 0.46
SLC6A2 P23975 1/20 0.41
BCAT2 O15382 1/20 0.40
ALDH1A1 P00352 3/20 0.40
MAPT P10636 2/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GRM6 O15303 1/20 0.38
ACHE P22303 1/20 0.37
BRS3 P32247 2/20 0.37
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
IDO1 P14902 2/20 0.36
LMNA P02545 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALOX12 P18054 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL517 0.87 SLC6A3 (0.50) SLC6A3SLC6A4SLC6A2BCAT2ALDH1A1
SCHEMBL9030773 0.81 CHRNB2 (0.45) SLC6A3SLC6A4ALDH1A1ACHEBRS3
Methylamine SCHEMBL28010440 0.80 BCAT2 (0.53) SLC6A3SLC6A4SLC6A2BCAT2ALDH1A1
SCHEMBL9531321 0.80 BCAT2 (0.52) SLC6A3SLC6A4SLC6A2BCAT2ALDH1A1
SCHEMBL29389473 0.80 BCAT2 (0.52) SLC6A3SLC6A4SLC6A2BCAT2ALDH1A1
SCHEMBL1665535 0.78 SLC6A3 (0.49) SLC6A3SLC6A4SLC6A2BCAT2ALDH1A1
Bromomethane SCHEMBL7011845 0.77 SLC6A3 (0.50) SLC6A3SLC6A4SLC6A2BCAT2ALDH1A1
SCHEMBL249 0.77 SLC6A3 (0.73) SLC6A3SLC6A4SLC6A2ALDH1A1MAPT
SCHEMBL3558536 0.76 SLC6A3 (0.48) SLC6A3SLC6A4SLC6A2BCAT2ACHE
SCHEMBL10533851 0.74 SLC6A3 (0.65) SLC6A3SLC6A4SLC6A2ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5336778-A Substituted triazoles as angiotensin II antagonists MERCK & CO., INC. (US) 1994-08-09 US disclosed
EP-0409332-A2 Substituted triazoles as angiotensin II antagonists MERCK & CO. INC. (US) 1991-01-23 EP disclosed