SCHEMBL9418908

SCHEMBL9418908

C=C(F)C(=O)OC(c1ccc(C)c(C)c1)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 2/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
LMNA P02545 3/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPK1 P28482 1/20 0.32
APP P05067 1/20 0.31
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
MAPT P10636 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
KIF11 P52732 2/20 0.31
TAS2R14 Q9NYV8 1/20 0.31
POLB P06746 1/20 0.30
CES2 O00748 1/20 0.30
CES1 P23141 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10396190 0.85 LMNA (0.38) LMNANPC1RAB9AMAPTNPSR1
SCHEMBL9418936 0.79 RORC (0.39) LMNAMAPK1NPC1RAB9AMAPT
SCHEMBL26794304 0.78 ESR1 (0.41) TDP1
SCHEMBL9418917 0.78 CA1 (0.36) LMNAMAPTNPSR1CES2CES1
SCHEMBL10396191 0.75 NPSR1 (0.37) LMNAKDM4EMAPTNPSR1CES2
SCHEMBL2465362 0.73 PGK1 (0.40) NPSR1L3MBTL1CES2SMN1; SMN2
SCHEMBL24908565 0.70 ESR1 (0.40) LMNAKDM4EMAPTNPSR1L3MBTL1
SCHEMBL7084775 0.70 RORC (0.38) LMNAMAPK1NPC1RAB9AMAPT
SCHEMBL26794329 0.70 ESR1 (0.32) LMNAMAPTNPSR1
SCHEMBL18857468 0.69 CYP19A1 (0.34) LMNANPC1RAB9AMAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5319131-A Reacting dimethyl 2-fluoromalonate with formaldehyde to form hydroxymethylated dimethyl 2-flurormalonate, hydrolysis, decarboxylation, dehydration then esterification with a hexafluoroalkylol HOECHST AKTIENGESELLSCHAFT (DE) 1994-06-07 US disclosed
US-5198925-A α-fluoroacrylic acid esters and polymers thereof HOECHST AKTIENGESELLSCHAFT 1993-03-30 US disclosed
EP-0203462-B1 ALPHA-FLUOROACRYLIC-ACID ESTERS AND THEIR POLYMERS HOECHST AKTIENGESELLSCHAFT (DE) 1990-08-01 EP disclosed
EP-0203462-A2 Alpha-fluoroacrylic-acid esters and their polymers HOECHST AKTIENGESELLSCHAFT (DE) 1986-12-03 EP disclosed