SCHEMBL9418917

SCHEMBL9418917

C=C(F)C(=O)OC(c1ccc(Br)cc1)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA5A P35218 1/20 0.36
CA9 Q16790 1/20 0.36
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CES2 O00748 2/20 0.31
CES1 P23141 2/20 0.31
OGG1 O15527 1/20 0.31
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
TSHR P16473 1/20 0.30
CYP2C19 P33261 1/20 0.30
ACHE P22303 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10396190 0.91 LMNA (0.38) LMNAMAPTNPSR1CES2CES1
SCHEMBL9418936 0.85 RORC (0.39) LMNAMAPTNPSR1CES2CES1
SCHEMBL9418908 0.78 PPARD (0.32) LMNAMAPTNPSR1CES2CES1
SCHEMBL10396191 0.77 NPSR1 (0.37) LMNAMAPTNPSR1CES2CES1
SCHEMBL24908565 0.72 ESR1 (0.40) LMNAMAPTNPSR1TSHR
SCHEMBL7084775 0.72 RORC (0.38) LMNAMAPTNPSR1
SCHEMBL15840364 0.71 SMN1; SMN2 (0.47) LMNANPSR1
SCHEMBL21834941 0.70 MAPT (0.40) CA1CA2CA5ACA9LMNA
SCHEMBL3692621 0.70 ELANE (0.41) LMNAMAPTNPSR1CES1CYP2D6
SCHEMBL9575390 0.69 LDHA (0.41) CA1CA2CA9LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5319131-A Reacting dimethyl 2-fluoromalonate with formaldehyde to form hydroxymethylated dimethyl 2-flurormalonate, hydrolysis, decarboxylation, dehydration then esterification with a hexafluoroalkylol HOECHST AKTIENGESELLSCHAFT (DE) 1994-06-07 US disclosed
US-5198925-A α-fluoroacrylic acid esters and polymers thereof HOECHST AKTIENGESELLSCHAFT 1993-03-30 US disclosed
EP-0203462-B1 ALPHA-FLUOROACRYLIC-ACID ESTERS AND THEIR POLYMERS HOECHST AKTIENGESELLSCHAFT (DE) 1990-08-01 EP disclosed
EP-0203462-A2 Alpha-fluoroacrylic-acid esters and their polymers HOECHST AKTIENGESELLSCHAFT (DE) 1986-12-03 EP disclosed