SCHEMBL9428375

SCHEMBL9428375

Cn1c(N2CCN(CCCOc3ccc(Cl)cc3C#N)CC2)cc(=O)n(C)c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
THRB P10828 1/20 0.43
HTR1A P08908 9/20 0.42
ADRA1B P35368 3/20 0.42
ADRA1A P35348 2/20 0.42
HTR2A P28223 7/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 2/20 0.41
LMNA P02545 2/20 0.41
ADRA1D P25100 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
FYN P06241 1/20 0.40
SRC P12931 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
DRD2 P14416 1/20 0.39
DRD3 P35462 1/20 0.39
TMEM97 Q5BJF2 1/20 0.39
SIGMAR1 Q99720 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9428300 0.88 DPP4 (0.43) ALDH1A1HTR1AADRA1BADRA1AHTR2A
SCHEMBL9429888 0.87 HTR1A (0.51) ALDH1A1HTR1AADRA1BADRA1AHTR2A
SCHEMBL9428509 0.86 HTR1A (0.40) ALDH1A1HTR1AADRA1BADRA1AHTR2A
SCHEMBL9387767 0.85 LMNA (0.52) ALDH1A1HTR1AADRA1BADRA1AHTR2A
SCHEMBL9428210 0.85 ADRA1B (0.47) ALDH1A1THRBHTR1AADRA1BADRA1A
SCHEMBL9428955 0.82 ALDH1A1 (0.45) ALDH1A1THRBHTR1AADRA1BADRA1A
SCHEMBL9429324 0.82 DRD2 (0.56) HTR1AHTR2ADRD2DRD3TMEM97
SCHEMBL9383816 0.81 KDM4E (0.47) ALDH1A1THRBHTR1AHTR2AMEN1
Oxalic Acid SCHEMBL9388735 0.81 LMNA (0.48) ALDH1A1HTR1AHTR2AMEN1KMT2A
Oxalic Acid SCHEMBL9388742 0.81 LMNA (0.48) ALDH1A1HTR1AHTR2AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5332739-A Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1994-07-26 US disclosed
EP-0454498-A2 Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1991-10-30 EP disclosed