SCHEMBL9428874

SCHEMBL9428874

Cn1c(N2CCN(CCCOc3ccc(C#N)cc3C(=O)c3ccccc3)CC2)cc(=O)n(C)c1=O

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 13/20 0.45
HRH3 Q9Y5N1 1/20 0.44
KCNA5 P22460 1/20 0.43
DRD2 P14416 1/20 0.42
DRD1 P21728 1/20 0.42
DRD3 P35462 1/20 0.42
HTR1A P08908 2/20 0.42
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 1/20 0.41
HTR2A P28223 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9428763 0.96 KCNA5 (0.48) HRH1KCNA5DRD2DRD1DRD3
SCHEMBL9429396 0.92 HRH3 (0.46) HRH1HRH3HTR1AHTR2A
SCHEMBL9429002 0.90 HRH3 (0.45) HRH1HRH3
SCHEMBL9428996 0.89 HRH3 (0.41) HRH1HRH3DRD2HTR1AADRA1D
SCHEMBL9428911 0.87 HRH1 (0.41) HRH1HRH3DRD2DRD3HTR1A
SCHEMBL9429278 0.84 HRH1 (0.45) HRH1KCNA5HTR1AADRA1DADRA1A
SCHEMBL9383925 0.84 ALDH1A1 (0.49) HRH1DRD2DRD1DRD3HTR1A
SCHEMBL9428459 0.84 KCNA5 (0.41) HRH1HRH3KCNA5DRD3HTR1A
SCHEMBL9429623 0.83 ALDH1A1 (0.48) HRH1KCNA5DRD2DRD3ADRA1D
SCHEMBL9428145 0.82 HRH1 (0.45) HRH1HRH3DRD2DRD1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5332739-A Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1994-07-26 US disclosed
EP-0454498-A2 Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1991-10-30 EP disclosed