SCHEMBL9433797

SCHEMBL9433797

O=C(C=Cc1ccccn1)Cc1cccnc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.51
MEN1 O00255 2/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
KMT2A Q03164 2/20 0.49
HTT P42858 1/20 0.47
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
HSP90AA1 P07900 1/20 0.44
CYP2D6 P10635 1/20 0.44
KDM4E B2RXH2 2/20 0.44
MAPT P10636 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
TBXAS1 P24557 2/20 0.44
ATM Q13315 1/20 0.42
POLB P06746 1/20 0.41
EPHX2 P34913 1/20 0.41
ERCC1 P07992 1/20 0.41
ERCC4 Q92889 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9433920 0.79 TBXAS1 (0.56) NAPRTMEN1NPC1RAB9AKMT2A
SCHEMBL9434718 0.79 NAPRT (0.50) NAPRTMEN1NPC1RAB9AKMT2A
SCHEMBL9434498 0.78 NAPRT (0.49) NAPRTKMT2AHTTCYP1A2CYP3A4
SCHEMBL9433799 0.78 MAPT (0.61) NAPRTMEN1NPC1RAB9AKMT2A
SCHEMBL9433617 0.78 HSD11B1 (0.50) NAPRTNPC1RAB9AKMT2ACYP1A2
SCHEMBL9433573 0.78 NAPRT (0.49) NAPRTNPC1RAB9AKMT2ACYP1A2
SCHEMBL9433826 0.77 TBXAS1 (0.57) NAPRTNPC1RAB9AKMT2AHTT
SCHEMBL9434219 0.77 ALDH1A1 (0.49) NAPRTMEN1NPC1RAB9AKMT2A
SCHEMBL9434333 0.77 RAB9A (0.60) NAPRTMEN1NPC1RAB9AKMT2A
SCHEMBL9433602 0.77 NAPRT (0.44) NAPRTCYP1A2CYP3A4CYP2C9CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed