SCHEMBL9449477

SCHEMBL9449477

c1ccc(COc2ccc3[nH]cc(C4CN5CCC4CC5)c3c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 2/20 0.52
NOS1 P29475 2/20 0.52
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C19 P33261 1/20 0.49
TRPM8 Q7Z2W7 2/20 0.49
KDM4E B2RXH2 1/20 0.49
MAPT P10636 1/20 0.49
LTA4H P09960 3/20 0.48
PLA2G2A P14555 3/20 0.48
CHRNB2 P17787 3/20 0.47
CHRNB4 P30926 3/20 0.47
CHRNA3 P32297 3/20 0.47
CHRNA7 P36544 3/20 0.47
CHRNA4 P43681 3/20 0.47
HTR1D P28221 3/20 0.47
ACHE P22303 1/20 0.46
SLC6A4 P31645 1/20 0.45
POLB P06746 1/20 0.44
MEN1 O00255 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9449311 0.92 IMPDH2 (0.50) NOS3NOS1CYP3A4CYP2C19TRPM8
SCHEMBL9448957 0.84 NOS3 (0.48) NOS3NOS1CYP3A4CYP2C19KDM4E
SCHEMBL9449109 0.83 HTR1A (0.47) NOS3NOS1CYP1A2CYP3A4CYP2C19
SCHEMBL9448836 0.81 HTR2A (0.61) NOS3NOS1SLC6A4
SCHEMBL9449668 0.79 TRPM8 (0.51) TRPM8KDM4EMAPTCHRNB2CHRNB4
SCHEMBL26863407 0.78 TRPM8 (0.56) CYP1A2CYP3A4CYP2C19TRPM8KDM4E
SCHEMBL5363538 0.78 CYP1A2 (0.60) NOS3NOS1CYP1A2CYP3A4CYP2C19
SCHEMBL4311896 0.77 HTR2C (0.55) NOS3NOS1CYP3A4CYP2C19KDM4E
SCHEMBL3546179 0.77 CYP3A4 (0.56) NOS3NOS1CYP1A2CYP3A4CYP2C19
SCHEMBL5705128 0.77 HTR2C (0.56) CYP1A2CYP3A4CYP2C19TRPM8KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5227386-A INDOLE DERIVATIVES MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1993-07-13 US disclosed