SCHEMBL9458372

SCHEMBL9458372

COC(=S)CCC(=O)Cc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
ALDH1A1 P00352 5/20 0.47
LMNA P02545 2/20 0.47
KDM4E B2RXH2 1/20 0.47
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
AKR1B1 P15121 1/20 0.44
RAB9A P51151 3/20 0.43
HPGD P15428 1/20 0.43
MAPT P10636 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
VNN1 O95497 1/20 0.43
TSHR P16473 1/20 0.42
NPC1 O15118 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7367260 0.86 CES2 (0.47) L3MBTL1TDP1ALDH1A1LMNAKDM4E
SCHEMBL490151 0.82 ALDH1A1 (0.68) L3MBTL1TDP1ALDH1A1LMNAKDM4E
SCHEMBL8619264 0.81 CES1 (0.64) L3MBTL1TDP1ALDH1A1LMNACES2
SCHEMBL7324968 0.79 ALDH1A1 (0.45) ALDH1A1LMNAKDM4ECES2CES1
SCHEMBL9457451 0.76 L3MBTL1 (0.44) L3MBTL1TDP1ALDH1A1LMNAKDM4E
SCHEMBL11062372 0.76 LMNA (0.59) L3MBTL1TDP1ALDH1A1LMNAKDM4E
SCHEMBL11067848 0.76 ALDH1A1 (0.44) L3MBTL1TDP1ALDH1A1LMNAKDM4E
SCHEMBL8620925 0.76 ALDH1A1 (0.61) L3MBTL1TDP1ALDH1A1KDM4ECES2
SCHEMBL8617001 0.76 TDP1 (0.58) L3MBTL1TDP1ALDH1A1CES2CES1
SCHEMBL2131696 0.75 AKR1B1 (0.62) L3MBTL1TDP1ALDH1A1LMNACES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5225421-A Leukotriene antagonists; cytoprotective agents MERCK FROSST CANADA, INC. (CA) 1993-07-06 US disclosed
EP-0275667-B1 3-HETERO-SUBSTITUTED-N-BENZYL-INDOLES MERCK FROSST CANADA INC. (CA) 1992-03-18 EP disclosed
US-5081138-A Antiasthmatic, antiallergic, antiinflammatory and cytoprotective agents MERCK FROSST CANADA, INC. (CA) 1992-01-14 US disclosed
EP-0275667-A1 3-hetero-substituted-N-benzyl-indoles MERCK FROSST CANADA INC. (CA) 1988-07-27 EP disclosed