SCHEMBL7324968

SCHEMBL7324968

COC(=S)Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.45
HPGD P15428 2/20 0.45
ALOX12 P18054 2/20 0.45
LMNA P02545 2/20 0.44
KDM4E B2RXH2 2/20 0.44
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
AKR1B1 P15121 1/20 0.44
KMT2A Q03164 3/20 0.44
GAA P10253 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
HTT P42858 1/20 0.44
RAB9A P51151 3/20 0.44
MAPT P10636 3/20 0.43
MEN1 O00255 2/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
POLB P06746 1/20 0.43
CYP3A4 P08684 1/20 0.43
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7367260 0.82 CES2 (0.47) ALDH1A1HPGDLMNAKDM4ECES2
SCHEMBL7632091 0.80 LMNA (0.49) ALDH1A1LMNAHTTIDO1
SCHEMBL9458372 0.79 L3MBTL1 (0.50) ALDH1A1HPGDLMNAKDM4ECES2
SCHEMBL3251246 0.78 ALDH1A1 (0.44) ALDH1A1LMNACES2CES1AKR1B1
SCHEMBL27791495 0.77 TSHR (0.61) ALOX12LMNACES2CES1AKR1B1
SCHEMBL29185461 0.77 CA12 (0.41) ALDH1A1ALOX12LMNACES2CES1
SCHEMBL9755852 0.77 IDO1 (0.43) ALDH1A1HPGDALOX12LMNACES2
SCHEMBL2154441 0.76 CES1 (0.48) ALDH1A1LMNAKDM4ECES2CES1
SCHEMBL6295378 0.76 CES2 (0.48) ALDH1A1LMNAKDM4ECES2CES1
SCHEMBL3048337 0.76 ALDH1A1 (0.59) ALDH1A1LMNACES2CES1AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691959-B1 HETEROCYCLIC DERIVATIVES AS PLATELET AGGREGATION INHIBITORS ZENECA LTD (GB) 1998-07-22 EP disclosed
EP-0825184-A1 Heterocyclic derivatives as platelet aggregation inhibitors ZENECA LIMITED (GB) 1998-02-25 EP disclosed
EP-0641207-A4 ENANTIOMERIC CYNEMICIN ANALOGS, PREPARATION AND USE THEREOF. SCRIPPS RESEARCH INST (US) 1996-08-14 EP disclosed
EP-0691959-A1 HETEROCYCLIC DERIVATIVES AS PLATELET AGGREGATION INHIBITORS ZENECA LIMITED (GB) 1996-01-17 EP disclosed
EP-0690847-A1 HETEROCYCLIC COMPOUNDS AS PLATELET AGGREGATION INHIBITORS ZENECA LIMITED (GB) 1996-01-10 EP disclosed
EP-0641207-A1 ENANTIOMERIC CYNEMICIN ANALOGS, PREPARATION AND USE THEREOF THE SCRIPPS RESEARCH INSTITUTE (US) 1995-03-08 EP disclosed
WO-1994022835-A2 HETEROCYCLIC COMPOUNDS AS PLATELET AGGREGATION INHIBITORS ZENECA LIMITED (GB) 1994-10-13 WO disclosed
WO-1994022834-A1 HETEROCYCLIC DERIVATIVES AS PLATELET AGGREGATION INHIBITORS ZENECA LIMITED (GB) 1994-10-13 WO disclosed
US-5281710-A Antibiotics or antitumor agents THE SCRIPPS RESEARCH INSTITUTE (US) 1994-01-25 US disclosed
WO-1993023046-A1 ENANTIOMERIC CYNEMICIN ANALOGS, PREPARATION AND USE THEREOF THE SCRIPPS RESEARCH INSTITUTE (US) 1993-11-25 WO disclosed
US-4980485-A Method of manufacturing optically-active periplanone-b JAPAN TOBACCO INC. (JP) 1990-12-25 US disclosed
US-4755626-A 4-isopropyl-7-methylene-5-cyclodecen-1-ol JAPAN TOBACCO, INC. (JP) 1988-07-05 US disclosed
US-4710581-A Nucleophilic substitution process ETHYL CORPORATION (US) 1987-12-01 US disclosed
US-4581463-A Nucleophilic substitution process combined with additional reaction steps ETHYL CORPORATION (US) 1986-04-08 US disclosed
US-RE29882-E SALT FORMATION, REARRANGEMENT, DESULFURIZATION OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 1979-01-16 US disclosed
US-4056569-A Ortho-[(alkylthio)(aminocarbonyl)methyl]anilines THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 1977-11-01 US disclosed
US-3996264-A Synthesis of oxindoles from anilines and intermediates therein THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 1976-12-07 US disclosed
US-3972894-A Synthesis of oxindoles from anilines and β-thio carboxylic esters or amides THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 1976-08-03 US disclosed