SCHEMBL9470388

SCHEMBL9470388

CC(C)N1C(=O)C(Sc2ccccc2)c2cccnc21

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.37
SRC P12931 1/20 0.32
MYC P01106 1/20 0.31
ALDH1A1 P00352 3/20 0.31
CCNA2 P20248 1/20 0.31
CDK2 P24941 1/20 0.31
HTT P42858 1/20 0.31
NPSR1 Q6W5P4 1/20 0.30
IDH1 O75874 1/20 0.30
MARK3 P27448 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9838569 0.82 SRC (0.41) TSHRSRCMYCALDH1A1CCNA2
SCHEMBL9470368 0.78 ALDH1A1 (0.43) ALDH1A1HTTNPSR1KMT2A
SCHEMBL9470466 0.78 KMT2A (0.47) TSHRALDH1A1HTTKMT2A
SCHEMBL9470397 0.77 ADRA2A (0.37) SRCALDH1A1CCNA2CDK2KMT2A
SCHEMBL9469978 0.75 LMNA (0.40) TSHRALDH1A1KMT2A
SCHEMBL4690229 0.73 ALDH1A1 (0.34) ALDH1A1KMT2A
SCHEMBL9469385 0.73 GAA (0.39) ALDH1A1KMT2A
SCHEMBL9470341 0.72 MEN1 (0.40) ALDH1A1HTTNPSR1KMT2A
SCHEMBL9469283 0.72 ALDH1A1 (0.39) TSHRALDH1A1HTTNPSR1KMT2A
SCHEMBL9470503 0.71 ALDH1A1 (0.40) ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5182289-A Pyrrolo 2,3-b!Pyridin-2-one Derivatives SCHERING CORPORATION (US) 1993-01-26 US claimed
EP-0419561-A1 HETEROBICYCLIC COMPOUNDS HAVING ANTIINFLAMMATORY ACTIVITY SCHERING CORPORATION (US) 1991-04-03 EP disclosed
WO-1989012637-A1 HETEROBICYCLIC COMPOUNDS HAVING ANTIINFLAMMATORY ACTIVITY SCHERING CORPORATION (US) 1989-12-28 WO disclosed