SCHEMBL9475698

SCHEMBL9475698

O=c1[nH]cnc2c1nnn2Cc1cccc(F)c1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.51
KMT2A Q03164 6/20 0.48
MEN1 O00255 5/20 0.48
HPGD P15428 5/20 0.48
POLB P06746 2/20 0.48
RAD51 Q06609 1/20 0.45
ROCK2 O75116 1/20 0.44
MAPT P10636 2/20 0.43
TSHR P16473 3/20 0.43
ALOX15 P16050 1/20 0.43
MMP13 P45452 1/20 0.43
TP53 P04637 1/20 0.43
ALDH1A1 P00352 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9476195 0.85 ADORA3 (0.51) KMT2AMEN1HPGDPOLBRAD51
SCHEMBL9475856 0.85 HPGD (0.59) GRM2KMT2AMEN1HPGDPOLB
SCHEMBL9477367 0.81 ADORA3 (0.46) KMT2AMEN1HPGDMAPTTSHR
SCHEMBL14094136 0.80 POLB (0.43) KMT2AMEN1HPGDPOLBRAD51
SCHEMBL9476624 0.78 TSHR (0.61) GRM2KMT2AMEN1HPGDPOLB
SCHEMBL9476484 0.75 GRM2 (0.53) GRM2KMT2AMEN1HPGDPOLB
SCHEMBL30931879 0.74 PDE8B (0.53) KMT2AMEN1HPGDTSHRALOX15
SCHEMBL9476371 0.72 LMNA (0.53) KMT2AMEN1HPGDTSHRTP53
SCHEMBL9476477 0.72 MEN1 (0.62) KMT2AMEN1HPGDTSHRTP53
SCHEMBL9478099 0.72 ALDH1A1 (0.56) GRM2HPGDMAPTTSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5204353-A 3-benzyl-3H-1,2,3-triazolo[4,5-d]pyrimidines, compositions thereof, and method of treating epilepsy therewith CIBA-GEIGY CORPORATION (US) 1993-04-20 US disclosed
EP-0288431-B1 3H-1,2,3-triazolo[4,5-d]pyrimidines CIBA-GEIGY AG (CH) 1992-08-19 EP disclosed
EP-0288431-A1 3H-1,2,3-triazolo[4,5-d]pyrimidines CIBA-GEIGY AG (CH) 1988-10-26 EP disclosed